Compile Data Set for Download or QSAR
Report error Found 100 Enz. Inhib. hit(s) with all data for entry = 50028349
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM23916(CHEMBL378657 | 3-amino-N-(3-{[(2S)-1-[4-(2-carbami...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257511(US8569313, 47 | CHEMBL498875 | (S)-methyl 4-(1-(2-...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257512(US8569313, 32 | CHEMBL444411 | (S)-4-(1-(2-(3-(3-a...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104914(CHEMBL507322 | US8569313, Inhibitor 26)
Affinity DataKi:  7.5nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257557(US8569313, 48 | CHEMBL492342 | (S)-4-(1-(2-(3-(3-a...)
Affinity DataKi:  12nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104911(CHEMBL493116 | US8569313, Inhibitor 23)
Affinity DataKi:  13nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257666((S)-3-amino-N-(3-(N-(1-(4-benzylpiperidin-1-yl)-3-...)
Affinity DataKi:  17nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104912(CHEMBL493936 | US8569313, Inhibitor 24)
Affinity DataKi:  31nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257663(US8569313, 55 | CHEMBL493117 | (S)-3-amino-N-(3-(N...)
Affinity DataKi:  33nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257664(US8569313, 54 | CHEMBL493118 | (S)-3-amino-N-(3-(N...)
Affinity DataKi:  37nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257665((S)-3-amino-N-(3-(N-(3-(3-carbamimidoylphenyl)-1-(...)
Affinity DataKi:  53nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257667((S)-4-(4-(2-(3-(3-aminopropanamido)phenylsulfonami...)
Affinity DataKi:  53nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104913(CHEMBL523865 | US8569313, Inhibitor 25)
Affinity DataKi:  65nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257761((R)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenyls...)
Affinity DataKi:  100nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257761((R)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenyls...)
Affinity DataKi:  100nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257665((S)-3-amino-N-(3-(N-(3-(3-carbamimidoylphenyl)-1-(...)
Affinity DataKi:  110nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257706((S)-3-amino-N-(3-(N-(3-(3-carbamimidoylphenyl)-1-(...)
Affinity DataKi:  150nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257707((R)-1-((S)-2-(3-(3-aminopropanamido)phenylsulfonam...)
Affinity DataKi:  180nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257510(CHEMBL495143 | US8569313, 49 | (S)-4-(1-(2-(3-(3-a...)
Affinity DataKi:  255nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257663(US8569313, 55 | CHEMBL493117 | (S)-3-amino-N-(3-(N...)
Affinity DataKi:  270nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257666((S)-3-amino-N-(3-(N-(1-(4-benzylpiperidin-1-yl)-3-...)
Affinity DataKi:  350nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257760(3-amino-N-(3-(N-((2S)-3-(3-carbamimidoylphenyl)-1-...)
Affinity DataKi:  395nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257760(3-amino-N-(3-(N-((2S)-3-(3-carbamimidoylphenyl)-1-...)
Affinity DataKi:  470nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257511(US8569313, 47 | CHEMBL498875 | (S)-methyl 4-(1-(2-...)
Affinity DataKi:  600nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257557(US8569313, 48 | CHEMBL492342 | (S)-4-(1-(2-(3-(3-a...)
Affinity DataKi:  670nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257512(US8569313, 32 | CHEMBL444411 | (S)-4-(1-(2-(3-(3-a...)
Affinity DataKi:  850nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257664(US8569313, 54 | CHEMBL493118 | (S)-3-amino-N-(3-(N...)
Affinity DataKi:  880nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104911(CHEMBL493116 | US8569313, Inhibitor 23)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104911(CHEMBL493116 | US8569313, Inhibitor 23)
Affinity DataKi:  1.25E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104914(CHEMBL507322 | US8569313, Inhibitor 26)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104912(CHEMBL493936 | US8569313, Inhibitor 24)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104914(CHEMBL507322 | US8569313, Inhibitor 26)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257512(US8569313, 32 | CHEMBL444411 | (S)-4-(1-(2-(3-(3-a...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM23916(CHEMBL378657 | 3-amino-N-(3-{[(2S)-1-[4-(2-carbami...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257664(US8569313, 54 | CHEMBL493118 | (S)-3-amino-N-(3-(N...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104912(CHEMBL493936 | US8569313, Inhibitor 24)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257557(US8569313, 48 | CHEMBL492342 | (S)-4-(1-(2-(3-(3-a...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257666((S)-3-amino-N-(3-(N-(1-(4-benzylpiperidin-1-yl)-3-...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257707((R)-1-((S)-2-(3-(3-aminopropanamido)phenylsulfonam...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257762((S)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenyls...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of matriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257706((S)-3-amino-N-(3-(N-(3-(3-carbamimidoylphenyl)-1-(...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257511(US8569313, 47 | CHEMBL498875 | (S)-methyl 4-(1-(2-...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257706((S)-3-amino-N-(3-(N-(3-(3-carbamimidoylphenyl)-1-(...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM104911(CHEMBL493116 | US8569313, Inhibitor 23)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257664(US8569313, 54 | CHEMBL493118 | (S)-3-amino-N-(3-(N...)
Affinity DataKi:  2.56E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257663(US8569313, 55 | CHEMBL493117 | (S)-3-amino-N-(3-(N...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257511(US8569313, 47 | CHEMBL498875 | (S)-methyl 4-(1-(2-...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257666((S)-3-amino-N-(3-(N-(1-(4-benzylpiperidin-1-yl)-3-...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasminogen(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257557(US8569313, 48 | CHEMBL492342 | (S)-4-(1-(2-(3-(3-a...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257665((S)-3-amino-N-(3-(N-(3-(3-carbamimidoylphenyl)-1-(...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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