Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50028378
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278373(2(R)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  27nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278305(2(R)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  46nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278071(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  52nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278817(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  83nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278072(2-(R,S)-{2-[(1-Methyl-1H-indole-2-carbonyl)-amino]...)
Affinity DataIC50:  92nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278816(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  288nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278135(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  445nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278199((2R,S)-3-(4-Benzyloxy-phenyl)-2-{2-[(1H-indole-2-c...)
Affinity DataIC50:  1.16E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278198((2R,S)-3-(4-Hydroxy-phenyl)-2-{2-[(1H-indole-2-car...)
Affinity DataIC50:  2.07E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278372(2(S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  2.75E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278248((1R,S)-1H-Indole-2-carboxylic acid [2-(1-methyl-2-...)
Affinity DataIC50:  3.15E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185259(2(R,S)-{2-[(1H-indole-2-carbonyl)amino]-benzoylami...)
Affinity DataIC50:  3.24E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278304(2-(S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylami...)
Affinity DataIC50:  4.64E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278815(CHEMBL498273 | {2-[(1H-Indole-2-carbonyl)-amino]-b...)
Affinity DataIC50:  5.52E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278200((1R,S)-1H-Indole-2-carboxylic acid [2-(1-carbamoyl...)
Affinity DataIC50:  8.53E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278373(2(R)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  1.14E+4nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Hartley guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278305(2(R)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  1.47E+4nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Hartley guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  1.64E+4nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Hartley guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278303(3-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  1.69E+4nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Hartley guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278816(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  2.74E+4nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Hartley guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed