Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50028489
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278141BDBM50278141((S)-N-(1-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]dec...)
Affinity DataIC50: 25nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 87188BDBM87188(N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 30nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278138BDBM50278138(N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 90nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278167BDBM50278167(N-(2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 110nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278141BDBM50278141((S)-N-(1-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]dec...)
Affinity DataIC50: 140nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278143BDBM50278143((S)-3,4-difluoro-N-(1-(4-oxo-1-phenyl-1,3,8-triaza...)
Affinity DataIC50: 150nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 87188BDBM87188(N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 150nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278143BDBM50278143((S)-3,4-difluoro-N-(1-(4-oxo-1-phenyl-1,3,8-triaza...)
Affinity DataIC50: 200nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278138BDBM50278138(N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 500nMAssay Description:Inhibition of PLD2 by biochemical assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 87185BDBM87185(cid_53470115 | 4-azanyl-3-methoxy-N-[2-(4-oxidanyl...)
Affinity DataIC50: 550nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 87187BDBM87187(N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 990nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278167BDBM50278167(N-(2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 87186BDBM87186(VU0364187-1 | N-[2-(4-oxo-1-phenyl-1,3,8-triazaspi...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278138BDBM50278138(N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 87186BDBM87186(VU0364187-1 | N-[2-(4-oxo-1-phenyl-1,3,8-triazaspi...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278142BDBM50278142((trans)-N-((S)-1-(4-oxo-1-phenyl-1,3,8-triazaspiro...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278172BDBM50278172((S)-3-methyl-N-(1-(4-oxo-1-phenyl-1,3,8-triazaspir...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026634BDBM50026634(1-(pyridin-2-yl)piperazine | 1-(2-pyridyl)piperazi...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50106393BDBM50106393(1-(pyridin-4-yl)piperazine | 1-Pyridin-4-yl-pipera...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 87187BDBM87187(N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 4.25E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 87185BDBM87185(cid_53470115 | 4-azanyl-3-methoxy-N-[2-(4-oxidanyl...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278171BDBM50278171(N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278138BDBM50278138(N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PLD1 by biochemical assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278137BDBM50278137((trans)-N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D1(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278137BDBM50278137((trans)-N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PLD1 in human Calu1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278171BDBM50278171(N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278172BDBM50278172((S)-3-methyl-N-(1-(4-oxo-1-phenyl-1,3,8-triazaspir...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase D2(Human)
Vanderbilt University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50278142BDBM50278142((trans)-N-((S)-1-(4-oxo-1-phenyl-1,3,8-triazaspiro...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of GFP-labeled PLD2 in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed