Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50038854
LigandChemical structure of BindingDB Monomer ID 50277487BDBM50277487(4alpha-Phorbol 12,13-dihexanoate | CHEMBL490470)
Affinity DataEC50:  70nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277491BDBM50277491(Lumi-4alpha-Phorbol 12,13-didecanoate | CHEMBL5049...)
Affinity DataEC50:  175nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50240777BDBM50240777(Decanoic acid (1aR,1bS,4aS,7aS,7bS,8R,9R,9aS)-9-de...)
Affinity DataEC50:  370nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50277486BDBM50277486(4alpha-Phorbol 13-decanoate | CHEMBL541720)
Affinity DataEC50:  450nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277490BDBM50277490(4alpha-Phorbol 12,13-dimyristate | CHEMBL451849)
Affinity DataEC50:  2.83E+3nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50057512BDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataEC50:  2.25E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277739BDBM50277739(4alpha-phorbol diacetate | CHEMBL484343)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277488BDBM50277488(4alpha-Phorbol 12,13-dioctanoate | CHEMBL507303)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277489BDBM50277489(4alpha-Phorbol 12,13-dinonanoate | CHEMBL130626)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277740BDBM50277740(4-Deoxy-4alpha-Phorbol 12,13-didecanoate | CHEMBL5...)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of mouse wild type TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed