Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 3219
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29500BDBM29500(Pyrazolo[1,5-a]-1,3,5-triazine, 13-25)
Affinity DataIC50: 1.60nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29505BDBM29505(Pyrazolo[1,5-a]-1,3,5-triazine, 13-30)
Affinity DataIC50: 2.40nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29488BDBM29488(Pyrazolo[1,5-a]-1,3,5-triazine, 13-13)
Affinity DataIC50: 3nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29499BDBM29499(Pyrazolo[1,5-a]-1,3,5-triazine, 13-24)
Affinity DataIC50: 3.10nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29489BDBM29489(Pyrazolo[1,5-a]-1,3,5-triazine, 13-14)
Affinity DataIC50: 3.10nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29493BDBM29493(Pyrazolo[1,5-a]-1,3,5-triazine, 13-18)
Affinity DataIC50: 3.5nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29492BDBM29492(Pyrazolo[1,5-a]-1,3,5-triazine, 13-17)
Affinity DataIC50: 4.5nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29504BDBM29504(Pyrazolo[1,5-a]-1,3,5-triazine, 13-29)
Affinity DataIC50: 4.90nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29494BDBM29494(Pyrazolo[1,5-a]-1,3,5-triazine, 13-19)
Affinity DataIC50: 5.10nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29496BDBM29496(Pyrazolo[1,5-a]-1,3,5-triazine, 13-21)
Affinity DataIC50: 5.70nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29490BDBM29490(Pyrazolo[1,5-a]-1,3,5-triazine, 13-15)
Affinity DataIC50: 6.10nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29498BDBM29498(Pyrazolo[1,5-a]-1,3,5-triazine, 13-23)
Affinity DataIC50: 6.60nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29491BDBM29491(Pyrazolo[1,5-a]-1,3,5-triazine, 13-16)
Affinity DataIC50: 7nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29503BDBM29503(Pyrazolo[1,5-a]-1,3,5-triazine, 13-28)
Affinity DataIC50: 8.10nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29497BDBM29497(Pyrazolo[1,5-a]-1,3,5-triazine, 13-22)
Affinity DataIC50: 8.5nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29495BDBM29495(Pyrazolo[1,5-a]-1,3,5-triazine, 13-20)
Affinity DataIC50: 12nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29482BDBM29482(Pyrazolo[1,5-a]-1,3,5-triazine, 13-7)
Affinity DataIC50: 12.8nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29483BDBM29483(Pyrazolo[1,5-a]-1,3,5-triazine, 13-8)
Affinity DataIC50: 13.8nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29487BDBM29487(Pyrazolo[1,5-a]-1,3,5-triazine, 13-12)
Affinity DataIC50: 14.5nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29480BDBM29480(Pyrazolo[1,5-a]-1,3,5-triazine, 13-5)
Affinity DataIC50: 14.9nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29502BDBM29502(Pyrazolo[1,5-a]-1,3,5-triazine, 13-27)
Affinity DataIC50: 17.6nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29486BDBM29486(Pyrazolo[1,5-a]-1,3,5-triazine, 13-11)
Affinity DataIC50: 23.8nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29485BDBM29485(Pyrazolo[1,5-a]-1,3,5-triazine, 13-10)
Affinity DataIC50: 24.8nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29476BDBM29476(Pyrazolo[1,5-a]-1,3,5-triazine, 13-1)
Affinity DataIC50: 25.6nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29481BDBM29481(Pyrazolo[1,5-a]-1,3,5-triazine, 13-6)
Affinity DataIC50: 32.8nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29479BDBM29479(Pyrazolo[1,5-a]-1,3,5-triazine, 13-4)
Affinity DataIC50: 58nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29501BDBM29501(Pyrazolo[1,5-a]-1,3,5-triazine, 13-26)
Affinity DataIC50: 81.6nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29484BDBM29484(Pyrazolo[1,5-a]-1,3,5-triazine, 13-9)
Affinity DataIC50: 91.9nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29478BDBM29478(Pyrazolo[1,5-a]-1,3,5-triazine, 13-3)
Affinity DataIC50: 133nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

LigandChemical structure of BindingDB Monomer ID 29477BDBM29477(Pyrazolo[1,5-a]-1,3,5-triazine, 13-2)
Affinity DataIC50: 1.00E+4nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2009
Entry Details Article
PubMed