Compile Data Set for Download or QSAR
Report error Found 138 Enz. Inhib. hit(s) with all data for entry = 50028647
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249662BDBM50249662(4'-(2-{[(2R)-2-(6-Aminopyridin-3-yl)-2-hydroxyethy...)
Affinity DataEC50:  0.0290nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249662BDBM50249662(4'-(2-{[(2R)-2-(6-Aminopyridin-3-yl)-2-hydroxyethy...)
Affinity DataEC50:  0.0290nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277527BDBM50277527((R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethyla...)
Affinity DataEC50:  0.0350nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277534BDBM50277534(3-(Cyclohexylamino)-4'-(2-{[(2R)-2-hydroxy-2-pyrid...)
Affinity DataEC50:  0.0620nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277526BDBM50277526((R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethyla...)
Affinity DataEC50:  0.0660nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249663BDBM50249663(4'-[2-[[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethy...)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277509BDBM50277509(3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-pyridin...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249640BDBM50249640(4'-(2-{[(2R)-2-(6-Aminopyridin-3-yl)-2-hydroxyethy...)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249640BDBM50249640(4'-(2-{[(2R)-2-(6-Aminopyridin-3-yl)-2-hydroxyethy...)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277530BDBM50277530(3-(Cyclohexylamino)-4'-(2-{[(2R)-2-hydroxy-2-pheny...)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249636BDBM50249636(4'-(2-{[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino}e...)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277525BDBM50277525((R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethyla...)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277533BDBM50277533(4'-(2-{[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino}e...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243112BDBM50243112(3-(Cyclohexyloxy)-4-(2-{[(2R)-2-hydroxy-2-(3-pyrid...)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243111BDBM50243111(4-(2-{[(2R)-2-Hydroxy-2-(3-pyridinyl)ethyl]amino}e...)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243112BDBM50243112(3-(Cyclohexyloxy)-4-(2-{[(2R)-2-hydroxy-2-(3-pyrid...)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236160BDBM50236160((R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-(...)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277536BDBM50277536(3-Cyclopentyl-4'-(2-{[(2R)-2-hydroxy-2-pyridin-3-y...)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236165BDBM50236165(3-(cyclohexyloxy)-4-(2-{[(2R)-2-hydroxy-2-phenylet...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277506BDBM50277506(4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-...)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277535BDBM50277535(4'-(2-{[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino}e...)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277480BDBM50277480(3-Cyclohexyl-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl]...)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236164BDBM50236164((R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-p...)
Affinity DataEC50:  0.340nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277505BDBM50277505(3-(Cycloheptyloxy)-4'-(2-{[(2R)-2-hydroxy-2-phenyl...)
Affinity DataEC50:  0.380nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277532BDBM50277532(3-Cyclopentyl-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl...)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277503BDBM50277503(3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-phenyle...)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277503BDBM50277503(3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-phenyle...)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236168BDBM50236168((R)-4'-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)...)
Affinity DataEC50:  0.460nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277531BDBM50277531(4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-...)
Affinity DataEC50:  0.460nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249638BDBM50249638(CHEMBL452134 | CHEMBL556852 | 4'-(2-{[(2R)-2-(4-Am...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249638BDBM50249638(CHEMBL452134 | CHEMBL556852 | 4'-(2-{[(2R)-2-(4-Am...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277507BDBM50277507(3-(Cyclohexylsulfanyl)-4'-(2-{[(2R)-2-hydroxy-2-ph...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277481BDBM50277481(3-(Cyclohexylmethyl)-4'-(2-{[(2R)-2-hydroxy-2-phen...)
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236184BDBM50236184(4-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}ethyl)-3...)
Affinity DataEC50:  0.560nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277529BDBM50277529(4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236181BDBM50236181(4-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}ethyl)-1...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277504BDBM50277504(4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277478BDBM50277478(3-(Cyclopentyloxy)-4'-(2-{[(2R)-2-hydroxy-2-phenyl...)
Affinity DataEC50:  0.620nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249639BDBM50249639(4'-(2-{[(2R)-2-(6-Aminopyridin-3-yl)-2-hydroxyethy...)
Affinity DataEC50:  0.680nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Dog)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277506BDBM50277506(4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-...)
Affinity DataEC50:  0.680nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Dog)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277503BDBM50277503(3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-phenyle...)
Affinity DataEC50:  0.830nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Dog)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277503BDBM50277503(3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-phenyle...)
Affinity DataEC50:  0.830nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25392BDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.840nMAssay Description:Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Dog)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277531BDBM50277531(4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-...)
Affinity DataEC50:  0.880nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25392BDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.970nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Dog)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249638BDBM50249638(CHEMBL452134 | CHEMBL556852 | 4'-(2-{[(2R)-2-(4-Am...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277508BDBM50277508(4'-(2-{[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino}e...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Dog)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277529BDBM50277529(4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236183BDBM50236183((R)-4'-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Dog)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236184BDBM50236184(4-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}ethyl)-3...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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