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Found 40 Enz. Inhib. hit(s) with all data for entry = 50028668
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259220(CHEMBL467091 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  49nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259134(CHEMBL466720 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  68nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259176(CHEMBL466257 | N-(3-(4-chlorobenzyl)-4-oxo-3,4-dih...)
Affinity DataIC50:  79nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259177(CHEMBL466674 | N-(3-(4-chloro-3-(trifluoromethyl)b...)
Affinity DataIC50:  110nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259217(CHEMBL512969 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  180nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259177(CHEMBL466674 | N-(3-(4-chloro-3-(trifluoromethyl)b...)
Affinity DataIC50:  190nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259088(CHEMBL466313 | benzyl 3-(3,4-dichlorobenzyl)-4-oxo...)
Affinity DataIC50:  193nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259220(CHEMBL467091 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  208nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259090(CHEMBL466314 | benzyl 3-(3-chloro-4-fluorobenzyl)-...)
Affinity DataIC50:  220nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259089(CHEMBL512775 | benzyl 3-(4-chlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  250nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259133(CHEMBL466719 | benzyl 3-(3,4-dimethylbenzyl)-4-oxo...)
Affinity DataIC50:  250nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259088(CHEMBL466313 | benzyl 3-(3,4-dichlorobenzyl)-4-oxo...)
Affinity DataIC50:  251nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259089(CHEMBL512775 | benzyl 3-(4-chlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  260nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259175(CHEMBL444433 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  261nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259134(CHEMBL466720 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  268nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259217(CHEMBL512969 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  348nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259133(CHEMBL466719 | benzyl 3-(3,4-dimethylbenzyl)-4-oxo...)
Affinity DataIC50:  790nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259090(CHEMBL466314 | benzyl 3-(3-chloro-4-fluorobenzyl)-...)
Affinity DataIC50:  865nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259261(2-(3-(3,4-dichlorobenzyl)-4-oxo-3,4-dihydroquinazo...)
Affinity DataIC50:  890nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259261(2-(3-(3,4-dichlorobenzyl)-4-oxo-3,4-dihydroquinazo...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259216(CHEMBL466885 | N-(3-(biphenyl-3-ylmethyl)-4-oxo-3,...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259087(CHEMBL467716 | benzyl 3-(3,4-dichlorobenzylcarbamo...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259176(CHEMBL466257 | N-(3-(4-chlorobenzyl)-4-oxo-3,4-dih...)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259178(2-hydroxy-N-(4-oxo-3-(3-(trifluoromethyl)benzyl)-3...)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259259(CHEMBL466889 | N-(3-(4-chlorobenzyl)-4-oxo-3,4-dih...)
Affinity DataIC50:  2.58E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259219(CHEMBL467090 | N-(3-(3-chlorobenzyl)-4-oxo-3,4-dih...)
Affinity DataIC50:  2.69E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259218(CHEMBL447081 | N-(3-(4-chlorobenzyl)-4-oxo-3,4-dih...)
Affinity DataIC50:  3.12E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259087(CHEMBL467716 | benzyl 3-(3,4-dichlorobenzylcarbamo...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259179(2-hydroxy-N-(4-oxo-3-(4-(trifluoromethyl)benzyl)-3...)
Affinity DataIC50:  3.42E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259216(CHEMBL466885 | N-(3-(biphenyl-3-ylmethyl)-4-oxo-3,...)
Affinity DataIC50:  3.85E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259260(CHEMBL466444 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  3.86E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259135(CHEMBL466524 | N-(3-(4-chlorobenzyl)-4-oxo-3,4-dih...)
Affinity DataIC50:  7.97E+3nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259331(CHEMBL466087 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Mus musculus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259175(CHEMBL444433 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of delta(5)-desaturase in mouse ABMC7 cells by high throughput radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Mus musculus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259087(CHEMBL467716 | benzyl 3-(3,4-dichlorobenzylcarbamo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of delta(5)-desaturase in mouse ABMC7 cells by high throughput radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259263((R)-N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4-dihydroqui...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259262((S)-N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4-dihydroqui...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Mus musculus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259175(CHEMBL444433 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of delta(6)-desaturase in mouse ABMC7 cells by high throughput radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259132(CHEMBL466522 | benzyl 3-(2,4-dichlorobenzyl)-4-oxo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of rat microsomal delta(9)-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Mus musculus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259087(CHEMBL467716 | benzyl 3-(3,4-dichlorobenzylcarbamo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of delta(6)-desaturase in mouse ABMC7 cells by high throughput radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed