Compile Data Set for Download or QSAR
maximum 50k data
Found 71 Enz. Inhib. hit(s) with all data for entry = 50028722
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278942(CHEMBL499905 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  80nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279256(CHEMBL527018 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  140nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278998(CHEMBL504926 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  190nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279026(CHEMBL505719 | rac-3-(1-benzyl-5-methoxy-2-methyl-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279256(CHEMBL527018 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  270nMAssay Description:Inhibition of MMP2 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279255(2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-methyl...)
Affinity DataIC50:  280nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279067(CHEMBL507022 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  280nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279110(CHEMBL498806 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  290nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278996(CHEMBL497904 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  300nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279071(CHEMBL503326 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  300nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279109(CHEMBL524912 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  320nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279152(CHEMBL525434 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  330nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279028(CHEMBL503835 | rac-3-(1-(benzo[d][1,3]dioxol-5-ylm...)
Affinity DataIC50:  330nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279108(CHEMBL499633 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  340nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279153(2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(3-cya...)
Affinity DataIC50:  410nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279154(CHEMBL500691 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  470nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279069(CHEMBL449253 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  490nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279068(CHEMBL504122 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  500nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278888(CHEMBL526567 | D-3-(1-(4-(allyloxy)benzyl)-1H-indo...)
Affinity DataIC50:  540nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279343(CHEMBL487755 | rac-3-(5-bromo-1H-indol-3-yl)-2-(4-...)
Affinity DataIC50:  630nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278997(CHEMBL525641 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  890nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279025(CHEMBL525730 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  900nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279416(CHEMBL452642 | D-3-(1-(biphenyl-2-ylmethyl)-1H-ind...)
Affinity DataIC50:  970nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278889(CHEMBL506243 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  980nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278974(CHEMBL524470 | L-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278995(CHEMBL497738 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279414(CHEMBL523616 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279257(2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-methox...)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of MMP2 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279377(CHEMBL487139 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  1.43E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278942(CHEMBL499905 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  1.44E+3nMAssay Description:Inhibition of MMP2 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279027(CHEMBL449262 | rac-3-(1-(benzo[d][1,3]dioxol-5-ylm...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279341(CHEMBL520686 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279375(CHEMBL487138 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279342(CHEMBL519909 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279413(CHEMBL520816 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  1.71E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279256(CHEMBL527018 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  1.81E+3nMAssay Description:Inhibition of MMP13 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278940(CHEMBL525428 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279415(CHEMBL483952 | D-3-(1-benzyl-1H-indol-3-yl)-2-(4-(...)
Affinity DataIC50:  2.15E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279070(CHEMBL507280 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  2.24E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279029(CHEMBL526385 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  2.24E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278913(CHEMBL502558 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279412(CHEMBL484617 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279221(CHEMBL498058 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  2.53E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279374(CHEMBL521238 | rac-2-(4-(but-2-ynyloxy)phenylsulfo...)
Affinity DataIC50:  2.96E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279287(3-(5-(benzyloxy)-1H-indol-3-yl)-2-(4-(but-2-ynylox...)
Affinity DataIC50:  3.27E+3nMAssay Description:Inhibition of MMP2 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278941(CHEMBL524677 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  3.45E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278915(CHEMBL501213 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  3.59E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279376(CHEMBL520548 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  3.67E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278914(CHEMBL524726 | D-2-(4-(but-2-ynyloxy)phenylsulfona...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279287(3-(5-(benzyloxy)-1H-indol-3-yl)-2-(4-(but-2-ynylox...)
Affinity DataIC50:  4.44E+3nMAssay Description:Inhibition of MMP13 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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