Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 3344
LigandChemical structure of BindingDB Monomer ID 31647BDBM31647(tetrahydrobenzothiophene (THBT), 21)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31648BDBM31648(tetrahydrobenzothiophene (THBT), 22)
Affinity DataIC50: 25nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31637BDBM31637(tetrahydrobenzothiophene (THBT), 6)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 31644BDBM31644(tetrahydrobenzothiophene (THBT), 23)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31638BDBM31638(tetrahydrobenzothiophene (THBT), 13a)
Affinity DataIC50: 79nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31649BDBM31649(tetrahydrobenzothiophene (THBT), 24)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31647BDBM31647(tetrahydrobenzothiophene (THBT), 21)
Affinity DataIC50: 126nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31648BDBM31648(tetrahydrobenzothiophene (THBT), 22)
Affinity DataIC50: 126nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31636BDBM31636(tetrahydrobenzothiophene (THBT), 4)
Affinity DataIC50: 200nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31636BDBM31636(tetrahydrobenzothiophene (THBT), 4)
Affinity DataIC50: 316nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31650BDBM31650(tetrahydrobenzothiophene (THBT), 25)
Affinity DataIC50: 398nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31644BDBM31644(tetrahydrobenzothiophene (THBT), 23)
Affinity DataIC50: 398nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31637BDBM31637(tetrahydrobenzothiophene (THBT), 6)
Affinity DataIC50: 501nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31640BDBM31640(tetrahydrobenzothiophene (THBT), 14)
Affinity DataIC50: 631nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31642BDBM31642(tetrahydrobenzothiophene (THBT), 16)
Affinity DataIC50: 1.26E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31646BDBM31646(tetrahydrobenzothiophene (THBT), 20)
Affinity DataIC50: 1.26E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31650BDBM31650(tetrahydrobenzothiophene (THBT), 25)
Affinity DataIC50: 1.59E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31645BDBM31645(tetrahydrobenzothiophene (THBT), 19)
Affinity DataIC50: 2.00E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31651BDBM31651(tetrahydrobenzothiophene (THBT), 18)
Affinity DataIC50: 2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31640BDBM31640(tetrahydrobenzothiophene (THBT), 14)
Affinity DataIC50: 2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31641BDBM31641(tetrahydrobenzothiophene (THBT), 15)
Affinity DataIC50: 2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31641BDBM31641(tetrahydrobenzothiophene (THBT), 15)
Affinity DataIC50: 2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31649BDBM31649(tetrahydrobenzothiophene (THBT), 24)
Affinity DataIC50: 2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31651BDBM31651(tetrahydrobenzothiophene (THBT), 18)
Affinity DataIC50: 5.01E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31643BDBM31643(tetrahydrobenzothiophene (THBT), 17)
Affinity DataIC50: 5.01E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31642BDBM31642(tetrahydrobenzothiophene (THBT), 16)
Affinity DataIC50: 6.31E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31645BDBM31645(tetrahydrobenzothiophene (THBT), 19)
Affinity DataIC50: 6.31E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31646BDBM31646(tetrahydrobenzothiophene (THBT), 20)
Affinity DataIC50: 6.31E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31639BDBM31639(tetrahydrobenzothiophene (THBT), 13b)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 31643BDBM31643(tetrahydrobenzothiophene (THBT), 17)
Affinity DataIC50: 3.16E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2009
Entry Details Article
PubMed