Affinity DataKi: 2.51nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.01nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 63.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 79.4nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 79.4nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.16E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: >5.01E+3nMAssay Description:Antagonist activity at human neuropeptide Y5 receptor expressed in HEK293 cells by FLIPR/Ca2+ methodMore data for this Ligand-Target Pair
Affinity DataKi: >6.31E+3nMAssay Description:Antagonist activity at human neuropeptide Y1 receptor expressed in CHO cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: >6.31E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: >6.31E+3nMAssay Description:Antagonist activity at human neuropeptide Y1 receptor expressed in CHO cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human neuropeptide Y5 receptor expressed in HEK293 cells by FLIPR/Ca2+ methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Antagonist activity at human neuropeptide Y2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity to neuropeptide Y2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Binding affinity to neuropeptide Y2 receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair