Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50030921
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataIC50:  1.01nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50304074(2-(2-methylquinolin-4-ylamino)-N-phenylacetamide |...)
Affinity DataIC50:  1.03nMAssay Description:Displacement of [3H]dynorphin from human kappa opioid receptor expressed in C6 giloma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50304074(2-(2-methylquinolin-4-ylamino)-N-phenylacetamide |...)
Affinity DataIC50:  1.15nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataIC50:  1.99nMAssay Description:Displacement of [3H]dynorphin from human kappa opioid receptor expressed in C6 giloma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed