Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50022598
TargetSerine/threonine-protein kinase PLK1(Human)
GlaxoSmithKline Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50355500(CHEMBL1908394 | US9695172, GSK461364)
Affinity DataKi: <0.5nMAssay Description:Time-dependent inhibition of full length human PLK1 assessed as apparent dissociation constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
GlaxoSmithKline Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50355500(CHEMBL1908394 | US9695172, GSK461364)
Affinity DataKi:  860nMAssay Description:Time-dependent inhibition of full length human PLK2 assessed as apparent dissociation constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
GlaxoSmithKline Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50355500(CHEMBL1908394 | US9695172, GSK461364)
Affinity DataKi:  1.00E+3nMAssay Description:Time-dependent inhibition of full length human PLK3 assessed as apparent dissociation constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed