Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50030714
TargetKappa-type opioid receptor(Human)
Biomedizinische Forschungsreagenzien

Curated by ChEMBL
LigandPNGBDBM50300442((20R)-4,5-alpha-Epoxy-17-methyl-3-hydroxy-6-methox...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]diprenorphine from human cloned kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Biomedizinische Forschungsreagenzien

Curated by ChEMBL
LigandPNGBDBM50300442((20R)-4,5-alpha-Epoxy-17-methyl-3-hydroxy-6-methox...)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]diprenorphine from human cloned mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Biomedizinische Forschungsreagenzien

Curated by ChEMBL
LigandPNGBDBM50300442((20R)-4,5-alpha-Epoxy-17-methyl-3-hydroxy-6-methox...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]naltrindole from human cloned delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed