Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50004484
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S/T165A mutantMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Inhibition of wild-type HIV1 Reverse transcriptaseMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of HIV1 Reverse transcriptase T165A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S mutantMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of HIV1 Reverse transcriptase T165A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Inhibition of HIV1 Reverse transcriptase M184V mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 370nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S/T165A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S/M184V mutantMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Inhibition of wild-type HIV1 Reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 640nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S/M184V mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 640nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 730nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S/T165A/M184V mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 790nMAssay Description:Inhibition of HIV1 Reverse transcriptase M184V mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Inhibition of HIV1 Reverse transcriptase P119S/T165A/M184V mutantMore data for this Ligand-Target Pair


3D Structure (crystal)