Compile Data Set for Download or QSAR
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Found 31 Enz. Inhib. hit(s) with all data for entry = 50030829
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50302304(1,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302299(2,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302303(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302295(CHEMBL570792 | N-(5-ethyl-4-(morpholinomethyl)pyri...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302302(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302305(2,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302301(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302300(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302294(2,2-dimethyl-N-(6-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302298(CHEMBL566456 | N-(5-methyl-4-(morpholinomethyl)pyr...)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302296(CHEMBL568157 | N-(5-cyano-4-(morpholinomethyl)pyri...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301314(2,2-dimethyl-N-(4-methyl-3-(morpholinomethyl)pheny...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301310(CHEMBL567924 | N-(2,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302297(CHEMBL572328 | N-(5-amino-4-(morpholinomethyl)pyri...)
Affinity DataKi:  870nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302302(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP55960 from human cloned CB1 receptor after 120 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302306(2,2-dimethyl-N-(5-methyl-6-(morpholinomethyl)pyrid...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302299(2,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]CP55960 from human cloned CB1 receptor after 120 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302304(1,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]CP55960 from human cloned CB1 receptor after 120 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302305(2,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [3H]CP55960 from human cloned CB1 receptor after 120 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302295(CHEMBL570792 | N-(5-ethyl-4-(morpholinomethyl)pyri...)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]CP55960 from human cloned CB1 receptor after 120 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302303(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataEC50:  8.80nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302304(1,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302305(2,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302298(CHEMBL566456 | N-(5-methyl-4-(morpholinomethyl)pyr...)
Affinity DataEC50:  70nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302301(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302302(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302300(1-ethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-...)
Affinity DataEC50:  62nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302295(CHEMBL570792 | N-(5-ethyl-4-(morpholinomethyl)pyri...)
Affinity DataEC50:  9.60nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302294(2,2-dimethyl-N-(6-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataEC50:  260nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302299(2,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302296(CHEMBL568157 | N-(5-cyano-4-(morpholinomethyl)pyri...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed