Compile Data Set for Download or QSAR
maximum 50k data
Found 86 Enz. Inhib. hit(s) with all data for entry = 50039090
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50378699(CHEMBL1204023)
Affinity DataIC50:  80nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50158453(CHEMBL224400 | N-(3-Phenylamino-4-pyridinyl)triflu...)
Affinity DataIC50:  90nMAssay Description:Inhibition of COX2 in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50158453(CHEMBL224400 | N-(3-Phenylamino-4-pyridinyl)triflu...)
Affinity DataIC50:  90nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311366(CHEMBL1079876 | N-[3-(4-methoxyphenylamino)-4-pyri...)
Affinity DataIC50:  100nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311392(CHEMBL1079335 | N-[3-(3-Bromophenylamino)-4-pyridi...)
Affinity DataIC50:  120nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50120981(1,1,1-trifluoro-N-(3-phenoxypyridin-4-yl)methanesu...)
Affinity DataIC50:  140nMAssay Description:Inhibition of COX1 in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311366(CHEMBL1079876 | N-[3-(4-methoxyphenylamino)-4-pyri...)
Affinity DataIC50:  160nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311396(CHEMBL1080231 | N-[3-(4-methylphenylamino)-4-pyrid...)
Affinity DataIC50:  170nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50158453(CHEMBL224400 | N-(3-Phenylamino-4-pyridinyl)triflu...)
Affinity DataIC50:  180nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50158453(CHEMBL224400 | N-(3-Phenylamino-4-pyridinyl)triflu...)
Affinity DataIC50:  180nMAssay Description:Inhibition of COX1 in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311389(CHEMBL1075636 | N-[3-(2-chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  190nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311398(CHEMBL1080405 | N-[3-(3-ethylphenylamino)-4-pyridi...)
Affinity DataIC50:  240nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311390(CHEMBL1077388 | N-[3-(3-Chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  270nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50378700(CHEMBL1204024)
Affinity DataIC50:  270nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50378699(CHEMBL1204023)
Affinity DataIC50:  330nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  350nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311391(CHEMBL1079333 | N-[3-(4-Chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  410nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50120980(CHEMBL148542 | N-(3-Phenoxy-pyridin-4-yl)-methanes...)
Affinity DataIC50:  410nMAssay Description:Inhibition of COX1 in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311395(CHEMBL1077403 | N-[3-(3-Methylphenylamino)-4-pyrid...)
Affinity DataIC50:  450nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311396(CHEMBL1080231 | N-[3-(4-methylphenylamino)-4-pyrid...)
Affinity DataIC50:  460nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311394(CHEMBL1081856 | N-[3-(2-methylphenylamino)-4-pyrid...)
Affinity DataIC50:  480nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311368(CHEMBL1079878 | N-[3-(2-chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  480nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311381(CHEMBL1078683 | N-[3-(4-methoxyphenylamino)-4-pyri...)
Affinity DataIC50:  560nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311373(CHEMBL1078374 | N-[3-(2-methylphenylamino)-4-pyrid...)
Affinity DataIC50:  560nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50120981(1,1,1-trifluoro-N-(3-phenoxypyridin-4-yl)methanesu...)
Affinity DataIC50:  620nMAssay Description:Inhibition of COX2 in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311398(CHEMBL1080405 | N-[3-(3-ethylphenylamino)-4-pyridi...)
Affinity DataIC50:  690nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50056999(CHEMBL56367 | nimesulide)
Affinity DataIC50:  700nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311369(CHEMBL1078090 | N-[3-(3-Chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  730nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311386(CHEMBL1079073 | N-(3-cycloheptylamino-4-pyridinyl)...)
Affinity DataIC50:  760nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311392(CHEMBL1079335 | N-[3-(3-Bromophenylamino)-4-pyridi...)
Affinity DataIC50:  910nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311399(CHEMBL1080406 | N-[3-(4-ethylphenylamino)-4-pyridi...)
Affinity DataIC50:  910nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311393(CHEMBL1081855 | N-[3-(4-bromophenylamino)-4-pyridi...)
Affinity DataIC50:  910nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50378701(CHEMBL1204025)
Affinity DataIC50:  940nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311395(CHEMBL1077403 | N-[3-(3-Methylphenylamino)-4-pyrid...)
Affinity DataIC50:  990nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311401(CHEMBL1079875 | N-[3-(3-methoxyphenylamino)-4-pyri...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311390(CHEMBL1077388 | N-[3-(3-Chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311400(CHEMBL1080407 | N-[3-(2-methoxyphenylamino)-4-pyri...)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311382(CHEMBL1078860 | N-(3-cyclopentylamino-4-pyridinyl)...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311391(CHEMBL1079333 | N-[3-(4-Chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50158452(CHEMBL224122 | N-(3-(phenylthio)pyridin-4-yl)metha...)
Affinity DataIC50:  1.19E+3nMAssay Description:Inhibition of COX2 in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311399(CHEMBL1080406 | N-[3-(4-ethylphenylamino)-4-pyridi...)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311370(CHEMBL1077398 | N-[3-(4-chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311375(CHEMBL1078376 | N-[3-(4-methylphenylamino)-4-pyrid...)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311401(CHEMBL1079875 | N-[3-(3-methoxyphenylamino)-4-pyri...)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311393(CHEMBL1081855 | N-[3-(4-bromophenylamino)-4-pyridi...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311386(CHEMBL1079073 | N-(3-cycloheptylamino-4-pyridinyl)...)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311388(CHEMBL1079074 | N-(3-phenylamino-4-pyridinyl)3,3,3...)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311389(CHEMBL1075636 | N-[3-(2-chlorophenylamino)-4-pyrid...)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of COX2 in LPS-stimulated human whole blood assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311372(CHEMBL1078373 | N-[3-(4-bromophenylamino)-4-pyridi...)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
University Of Liege

Curated by ChEMBL
LigandPNGBDBM50311367(CHEMBL1079877 | N-(3-phenylamino-4-pyridinyl)metha...)
Affinity DataIC50:  2.26E+3nMAssay Description:Inhibition of COX1 in human whole blood assessed as TXB2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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