Compile Data Set for Download or QSAR
Report error Found 140 Enz. Inhib. hit(s) with all data for entry = 3454
TargetSerine/threonine-protein kinase pim-3(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35048BDBM35048(benzothienopyrimidinone deriv., 20c)
Affinity DataKi:  0.400nM ΔG°:  -53.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35042BDBM35042(benzothienopyrimidinone deriv., 18b)
Affinity DataKi:  0.600nM ΔG°:  -52.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35048BDBM35048(benzothienopyrimidinone deriv., 20c)
Affinity DataKi:  0.700nM ΔG°:  -52.3kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35050BDBM35050(benzothienopyrimidinone deriv., 20e)
Affinity DataKi:  0.800nM ΔG°:  -51.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35043BDBM35043(benzothienopyrimidinone deriv., 19a)
Affinity DataKi:  0.800nM ΔG°:  -51.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 34997BDBM34997(benzothienopyrimidinone deriv., 6n)
Affinity DataKi:  0.900nM ΔG°:  -51.3kJ/molepH: 7.5 T: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35050BDBM35050(benzothienopyrimidinone deriv., 20e)
Affinity DataKi:  0.900nM ΔG°:  -51.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35012BDBM35012(benzothienopyrimidinone deriv., 12b)
Affinity DataKi:  1nM ΔG°:  -51.0kJ/molepH: 7.5 T: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35021BDBM35021(benzothienopyrimidinone deriv., 14f)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35041BDBM35041(benzothienopyrimidinone deriv., 18a)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35028BDBM35028(benzothienopyrimidinone deriv., 14m)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35033BDBM35033(benzothienopyrimidinone deriv., 15a)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35037BDBM35037(benzothienopyrimidinone deriv., 16a)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35048BDBM35048(benzothienopyrimidinone deriv., 20c)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35041BDBM35041(benzothienopyrimidinone deriv., 18a)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35026BDBM35026(benzothienopyrimidinone deriv., 14k)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35025BDBM35025(benzothienopyrimidinone deriv., 14j)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35026BDBM35026(benzothienopyrimidinone deriv., 14k)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35044BDBM35044(benzothienopyrimidinone deriv., 19b)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35045BDBM35045(benzothienopyrimidinone deriv., 19c)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35012BDBM35012(benzothienopyrimidinone deriv., 12b)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35015BDBM35015(benzothienopyrimidinone deriv., 13c)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35031BDBM35031(benzothienopyrimidinone deriv., 14p)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35034BDBM35034(benzothienopyrimidinone deriv., 15b)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35019BDBM35019(benzothienopyrimidinone deriv., 14d)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35037BDBM35037(benzothienopyrimidinone deriv., 16a)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35046BDBM35046(benzothienopyrimidinone deriv., 20a)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35025BDBM35025(benzothienopyrimidinone deriv., 14j)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35047BDBM35047(benzothienopyrimidinone deriv., 20b)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35049BDBM35049(benzothienopyrimidinone deriv., 20d)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35016BDBM35016(benzothienopyrimidinone deriv., 14a)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35032BDBM35032(benzothienopyrimidinone deriv., 14q)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35033BDBM35033(benzothienopyrimidinone deriv., 15a)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35021BDBM35021(benzothienopyrimidinone deriv., 14f)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35039BDBM35039(benzothienopyrimidinone deriv., 17a)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35029BDBM35029(benzothienopyrimidinone deriv., 14n)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35020BDBM35020(benzothienopyrimidinone deriv., 14e)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35039BDBM35039(benzothienopyrimidinone deriv., 17a)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 34988BDBM34988(benzothienopyrimidinone deriv., 6e)
Affinity DataKi:  5nM ΔG°:  -47.1kJ/molepH: 7.5 T: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35023BDBM35023(benzothienopyrimidinone deriv., 14h)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35005BDBM35005(benzothienopyrimidinone deriv., 8)
Affinity DataKi:  5nM ΔG°:  -47.1kJ/molepH: 7.5 T: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35024BDBM35024(benzothienopyrimidinone deriv., 14i)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35028BDBM35028(benzothienopyrimidinone deriv., 14m)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35046BDBM35046(benzothienopyrimidinone deriv., 20a)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35013BDBM35013(benzothienopyrimidinone deriv., 13a)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35035BDBM35035(benzothienopyrimidinone deriv., 15c)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35018BDBM35018(benzothienopyrimidinone deriv., 14c)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35042BDBM35042(benzothienopyrimidinone deriv., 18b)
Affinity DataKi:  6nM ΔG°:  -46.9kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35036BDBM35036(benzothienopyrimidinone deriv., 15d)
Affinity DataKi:  7nM ΔG°:  -46.5kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 35030BDBM35030(benzothienopyrimidinone deriv., 14o)
Affinity DataKi:  8nM ΔG°:  -46.2kJ/moleT: 2°CAssay Description:In 384-well v-bottom polypropylene plates, compound (2% DMSO) was mixed with Pim kinase and peptide substrate, followed by immediate initiation with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2009
Entry Details Article
PubMed
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