Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50030678
TargetEpidermal growth factor receptor(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 9nMAssay Description:Inhibition of Her1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 13nMAssay Description:Inhibition of Her1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 18nMAssay Description:Inhibition of Her2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM5445(N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(...)
Affinity DataIC50: 36nMAssay Description:Inhibition of Her2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 42nMAssay Description:Inhibition of Her2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM5445(N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(...)
Affinity DataIC50: 52nMAssay Description:Inhibition of Her1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Her4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 100nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 100nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Abl1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 100nMAssay Description:Inhibition of RetMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Her4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 300nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Abl1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 600nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 700nMAssay Description:Inhibition of RetMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Her1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Her2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of FGFR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of Flt4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of FGFR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of Flt4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MAPK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDGFRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Flt3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MetMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of KitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetInsulin-like growth factor 1 receptor(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MAPK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Raf1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300027((S)-1-Acryloyl-N-[4-(3-chloro-2,4-difluorophenylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Flt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Raf1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDGFRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Flt3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Flt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MetMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Hanmi Research Center

Curated by ChEMBL
LigandPNGBDBM50300026((S)-1-Acryloyl-N-[4-(3-chloro-2-fluorophenylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
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