Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 4814
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82141(WIN 55212-2)
Affinity DataKi:  7.30nM ΔG°:  -46.4kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82135(5-Substituted derivative, 5)
Affinity DataKi:  8.40nM ΔG°:  -46.1kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82140(4-methyl-N-({1-[2-(morpholin-4-yl)ethyl]-1H-indol-...)
Affinity DataKi:  15.7nM ΔG°:  -44.5kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82139(4-chloro-N-({1-[2-(morpholin-4-yl)ethyl]-1H-indol-...)
Affinity DataKi:  24.1nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82137(4-methoxy-N-({1-[2-(morpholin-4-yl)ethyl]-1H-indol...)
Affinity DataKi:  42.6nM ΔG°:  -42.1kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82138(N-({1-[2-(morpholin-4-yl)ethyl]-1H-indol-3-yl}meth...)
Affinity DataKi:  49.4nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82136(5-Substituted derivative, 6)
Affinity DataKi:  69.6nM ΔG°:  -40.9kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82132(5-Substituted derivative, 2)
Affinity DataKi:  74.6nM ΔG°:  -40.7kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82131(3-(Arylimino)-1-(2-morpholin-4-yl-ethyl)-1,3-dihyd...)
Affinity DataKi:  311nM ΔG°:  -37.1kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82133(5-Substituted derivative, 3)
Affinity DataKi:  390nM ΔG°:  -36.6kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
UniversitÀ

LigandPNGBDBM82134(3-(Arylimino)-1-(2-morpholin-4-yl-ethyl)-1,3-dihyd...)
Affinity DataKi:  553nM ΔG°:  -35.7kJ/molepH: 7.4 T: 2°CAssay Description:CB1 competitive assay were performed in rat cerebellar membranes using [3H]WIN 55212-2 from Perkin-Elmer as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed