Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50041758
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414981BDBM50414981(CHEMBL567417)
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414959BDBM50414959(CHEMBL409224)
Affinity DataIC50: 2.51nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414974BDBM50414974(CHEMBL568523)
Affinity DataIC50: 2.63nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414982BDBM50414982(CHEMBL579072)
Affinity DataIC50: 2.63nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414980BDBM50414980(CHEMBL568294)
Affinity DataIC50: 2.82nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414983BDBM50414983(CHEMBL574655)
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414986BDBM50414986(CHEMBL568522)
Affinity DataIC50: 5.62nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414958BDBM50414958(CHEMBL259243)
Affinity DataIC50: 6.46nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414975BDBM50414975(CHEMBL584087)
Affinity DataIC50: 6.61nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414978BDBM50414978(CHEMBL566543)
Affinity DataIC50: 8.13nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414964BDBM50414964(CHEMBL271128)
Affinity DataIC50: 11.5nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414966BDBM50414966(CHEMBL573216)
Affinity DataIC50: 14.8nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414967BDBM50414967(CHEMBL271801)
Affinity DataIC50: 17.4nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414957BDBM50414957(CHEMBL429436)
Affinity DataIC50: 19.1nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414977BDBM50414977(CHEMBL567627)
Affinity DataIC50: 22.4nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414976BDBM50414976(CHEMBL566324)
Affinity DataIC50: 22.4nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414968BDBM50414968(CHEMBL410885)
Affinity DataIC50: 27.5nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414964BDBM50414964(CHEMBL271128)
Affinity DataIC50: 30.2nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414979BDBM50414979(CHEMBL583621)
Affinity DataIC50: 30.9nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414969BDBM50414969(CHEMBL272022)
Affinity DataIC50: 32.4nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414959BDBM50414959(CHEMBL409224)
Affinity DataIC50: 34.7nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414964BDBM50414964(CHEMBL271128)
Affinity DataIC50: 45.7nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414970BDBM50414970(CHEMBL583843)
Affinity DataIC50: 55.0nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414962BDBM50414962(CHEMBL566759)
Affinity DataIC50: 70.8nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414966BDBM50414966(CHEMBL573216)
Affinity DataIC50: 70.8nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414957BDBM50414957(CHEMBL429436)
Affinity DataIC50: 81.3nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414958BDBM50414958(CHEMBL259243)
Affinity DataIC50: 81.3nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414958BDBM50414958(CHEMBL259243)
Affinity DataIC50: 83.2nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414959BDBM50414959(CHEMBL409224)
Affinity DataIC50: 87.1nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414971BDBM50414971(CHEMBL567202)
Affinity DataIC50: 95.5nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414961BDBM50414961(CHEMBL567419)
Affinity DataIC50: 107nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414965BDBM50414965(CHEMBL270971)
Affinity DataIC50: 115nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414966BDBM50414966(CHEMBL573216)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414972BDBM50414972(CHEMBL568296)
Affinity DataIC50: 129nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414960BDBM50414960(CHEMBL567620)
Affinity DataIC50: 141nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414984BDBM50414984(CHEMBL566974)
Affinity DataIC50: 141nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414965BDBM50414965(CHEMBL270971)
Affinity DataIC50: 209nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414965BDBM50414965(CHEMBL270971)
Affinity DataIC50: 219nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414984BDBM50414984(CHEMBL566974)
Affinity DataIC50: 229nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414967BDBM50414967(CHEMBL271801)
Affinity DataIC50: 363nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414967BDBM50414967(CHEMBL271801)
Affinity DataIC50: 447nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414963BDBM50414963(CHEMBL583212)
Affinity DataIC50: 525nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414957BDBM50414957(CHEMBL429436)
Affinity DataIC50: 603nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414975BDBM50414975(CHEMBL584087)
Affinity DataIC50: 759nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414962BDBM50414962(CHEMBL566759)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414968BDBM50414968(CHEMBL410885)
Affinity DataIC50: 1.41E+3nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414973BDBM50414973(CHEMBL572537)
Affinity DataIC50: 1.48E+3nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50414985BDBM50414985(CHEMBL568503)
Affinity DataIC50: 1.82E+3nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414961BDBM50414961(CHEMBL567419)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50414983BDBM50414983(CHEMBL574655)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
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