Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50031384
TargetM-phase inducer phosphatase 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM15190(3-(5-{[(5E)-2-amino-3,7-dicyano-4,6-dimethyl-5H-cy...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of recombinant MBP tagged CDC25B assessed as substrate 3-O-methylfluorescein fluorescent emission after 4 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50312523((E)-2-amino-5-(4-hydroxybenzylidene)-4,6-dimethyl-...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of "N-terminal GST-tagged human B-Raf assessed as luminescence activity after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM15190(3-(5-{[(5E)-2-amino-3,7-dicyano-4,6-dimethyl-5H-cy...)
Affinity DataIC50: 6.02E+4nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM15189(4-(5-{[(5E)-2-amino-3,7-dicyano-4,6-dimethyl-5H-cy...)
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed