Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50031205
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-((3,5-dichlorophenyl)carbamothioyl)piperazin-...)
Affinity DataKi:  1.90E+3nMAssay Description:Competitive-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-((9H-xanthene-9-carbonyl)carbamothioyl)pipera...)
Affinity DataKi:  2.70E+3nMAssay Description:Competitive-type inhibition of autotaxin-mediated pNP-TMP hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-((9H-xanthene-9-carbonyl)carbamothioyl)pipera...)
Affinity DataKi:  2.70E+3nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308959(4,4'-(5,5'-carbonylbis(1,3-dioxoisoindoline-5,2-di...)
Affinity DataKi:  5.00E+3nMAssay Description:Competitive-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308958(4-(4-(2-(naphthalen-1-yl)-1,3-dioxoisoindoline-5-c...)
Affinity DataKi:  5.80E+3nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308961(4-(2-(3-ethyl-4-oxo-3,4,6,7,8,9-hexahydropyrimido[...)
Affinity DataKi:  6.50E+3nMAssay Description:Noncompetitive inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-((3,5-dichlorophenyl)carbamothioyl)piperazin-...)
Affinity DataKi:  6.50E+3nMAssay Description:Noncompetitive inhibition of autotaxin-mediated pNP-TMP hydrolysis by Michaelis-Menton analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-((3,5-dichlorophenyl)carbamothioyl)piperazin-...)
Affinity DataKi:  6.50E+3nMAssay Description:Noncompetitive inhibition of autotaxin-mediated pNP-TMP hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308961(4-(2-(3-ethyl-4-oxo-3,4,6,7,8,9-hexahydropyrimido[...)
Affinity DataKi:  9.30E+3nMAssay Description:Noncompetitive inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308957(3-(1,3-dioxo-2-(4-(phenyldiazenyl)phenyl)isoindoli...)
Affinity DataKi:  1.51E+4nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-((9H-xanthene-9-carbonyl)carbamothioyl)pipera...)
Affinity DataKi:  1.98E+4nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308958(4-(4-(2-(naphthalen-1-yl)-1,3-dioxoisoindoline-5-c...)
Affinity DataKi:  3.23E+4nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308957(3-(1,3-dioxo-2-(4-(phenyldiazenyl)phenyl)isoindoli...)
Affinity DataKi:  4.03E+4nMAssay Description:Mixed-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menton analysis for enzyme-substrate complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-((3,5-dichlorophenyl)carbamothioyl)piperazin-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of autotaxin-mediated pNP-TMP hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-((9H-xanthene-9-carbonyl)carbamothioyl)pipera...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50300214(2-(4-((3,5-dichlorophenyl)carbamothioyl)piperazin-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308961(4-(2-(3-ethyl-4-oxo-3,4,6,7,8,9-hexahydropyrimido[...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308960(2-(4-((9H-xanthene-9-carbonyl)carbamothioyl)pipera...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of autotaxin-mediated pNP-TMP hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308958(4-(4-(2-(naphthalen-1-yl)-1,3-dioxoisoindoline-5-c...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of autotaxin-mediated pNP-TMP hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308958(4-(4-(2-(naphthalen-1-yl)-1,3-dioxoisoindoline-5-c...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308957(3-(1,3-dioxo-2-(4-(phenyldiazenyl)phenyl)isoindoli...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50308959(4,4'-(5,5'-carbonylbis(1,3-dioxoisoindoline-5,2-di...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells by amplex red protocolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed