Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 8086
TargetProthrombin(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233008(H-D-Ser-Ala-Arg-NH-(CH2)8-NH2 (7))
Affinity DataKi:  240nMpH: 8.4Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233006(H-D-Ser-Ala-Arg-NH-(CH2)6-NH2 (5))
Affinity DataKi:  2.50E+3nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233009(H-D-Ser-Ala-Arg-NH-(CH2)9-NH2 (8))
Affinity DataKi:  5.00E+3nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233005(H-D-Ser-Ala-Arg-NH-(CH2)5-NH2 (4))
Affinity DataKi:  6.30E+3nMpH: 8.8Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233012(H-D-Ser-Ala-Arg-NH-(CH2)4-OH (11))
Affinity DataKi:  1.00E+4nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233008(H-D-Ser-Ala-Arg-NH-(CH2)8-NH2 (7))
Affinity DataKi:  1.00E+4nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233011(H-D-Ser-Ala-Arg-NH-(CH2)3-OH (10))
Affinity DataKi:  1.50E+4nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233007(H-D-Ser-Ala-Arg-NH-(CH2)7-NH2 (6))
Affinity DataKi:  3.00E+4nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233005(H-D-Ser-Ala-Arg-NH-(CH2)5-NH2 (4))
Affinity DataKi:  3.70E+4nMpH: 7.4Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233008(H-D-Ser-Ala-Arg-NH-(CH2)8-NH2 (7))
Affinity DataKi:  8.70E+4nMpH: 8.8Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233009(H-D-Ser-Ala-Arg-NH-(CH2)9-NH2 (8))
Affinity DataKi:  9.00E+4nMpH: 7.4Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233006(H-D-Ser-Ala-Arg-NH-(CH2)6-NH2 (5))
Affinity DataKi:  1.81E+5nMpH: 7.4Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233007(H-D-Ser-Ala-Arg-NH-(CH2)7-NH2 (6))
Affinity DataKi:  2.44E+5nMpH: 8.8Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233009(H-D-Ser-Ala-Arg-NH-(CH2)9-NH2 (8))
Affinity DataKi:  2.93E+5nMpH: 8.8Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233007(H-D-Ser-Ala-Arg-NH-(CH2)7-NH2 (6))
Affinity DataKi:  3.64E+5nMpH: 7.4Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233012(H-D-Ser-Ala-Arg-NH-(CH2)4-OH (11))
Affinity DataKi:  5.45E+5nMpH: 7.4Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233010(H-D-Ser-Ala-Arg-NH-(CH2)2-OH (9))
Affinity DataKi:  7.27E+5nMpH: 7.4Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233011(H-D-Ser-Ala-Arg-NH-(CH2)3-OH (10))
Affinity DataKi:  1.09E+6nMpH: 7.4Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed