Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50039077
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50172158((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309538(5-Ethyl-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  1.03nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309540(2-Ethyl-5-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309534(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309537(2,5-dimethyl-1-phenyl-N-(2-(trifluoromethyl)benzyl...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309543(5-Bromo-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309536(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309539(5-Butyl-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309544(2-Methyl-5-methylsulfanyl-1-phenyl-1H-imidazole-4-...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309541(2-Ethyl-1-phenyl-1H-imidazole-4-carboxylic acid ad...)
Affinity DataKi:  12.7nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309535(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  13.8nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309546(1-Cyclohexyl-2,5-dimethyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309533(CHEMBL599070 | N-(((cis)-6,6-dimethylbicyclo[3.1.1...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309542(5-Chloro-2-methyl-1-phenyl-1H-imidazole-4-carboxyl...)
Affinity DataKi:  23.8nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309545(2,5-Dichloro-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM85739(CHEMBL178372 | JTE-907 | N-(1,3-Benzodioxole-5-ylm...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309532(CHEMBL603476 | N-(((cis)-6,6-dimethylbicyclo[3.1.1...)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309545(2,5-Dichloro-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309541(2-Ethyl-1-phenyl-1H-imidazole-4-carboxylic acid ad...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309537(2,5-dimethyl-1-phenyl-N-(2-(trifluoromethyl)benzyl...)
Affinity DataKi:  1.42E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309539(5-Butyl-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309535(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  3.01E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50172158((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  3.54E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM85739(CHEMBL178372 | JTE-907 | N-(1,3-Benzodioxole-5-ylm...)
Affinity DataKi:  3.92E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309533(CHEMBL599070 | N-(((cis)-6,6-dimethylbicyclo[3.1.1...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309540(2-Ethyl-5-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  4.15E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309534(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  4.89E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309536(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  5.44E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309544(2-Methyl-5-methylsulfanyl-1-phenyl-1H-imidazole-4-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309538(5-Ethyl-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309532(CHEMBL603476 | N-(((cis)-6,6-dimethylbicyclo[3.1.1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309546(1-Cyclohexyl-2,5-dimethyl-1H-imidazole-4-carboxyli...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309543(5-Bromo-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309542(5-Chloro-2-methyl-1-phenyl-1H-imidazole-4-carboxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed