Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50031262
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50310096((7,12-dihydro-3-methoxytetraphen-12-yl)methanamine...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]Ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50310098(N-((9,10-Dihydroanthracen-9-yl)methyl)-3-phenylpro...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]Ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50310097(N-((9,10-Dihydroanthracen-9-yl)methyl)-2-phenyleth...)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]Pyrilamine from human cloned histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50310099(N-((9,10-Dihydroanthracen-9-yl)methyl)-4-phenylbut...)
Affinity DataKi:  365nMAssay Description:Displacement of [3H]Ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50310097(N-((9,10-Dihydroanthracen-9-yl)methyl)-2-phenyleth...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]Ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50097644(9-(N-benzylaminomethyl)-9,10-dihydroanthracene | B...)
Affinity DataKi:  721nMAssay Description:Displacement of [3H]Ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50310098(N-((9,10-Dihydroanthracen-9-yl)methyl)-3-phenylpro...)
Affinity DataKi:  725nMAssay Description:Displacement of [3H]Pyrilamine from human cloned histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50310099(N-((9,10-Dihydroanthracen-9-yl)methyl)-4-phenylbut...)
Affinity DataKi:  964nMAssay Description:Displacement of [3H]Pyrilamine from human cloned histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50310096((7,12-dihydro-3-methoxytetraphen-12-yl)methanamine...)
Affinity DataKi:  2.64E+3nMAssay Description:Displacement of [3H]Pyrilamine from human cloned histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed