Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50031272
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5447BDBM5447(ZD1839 | N-(3-chloro-4-fluorophenyl)-7-methoxy-6-[...)
Affinity DataIC50: 33nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310276BDBM50310276(N-Hexadecyl 2-(5-hydroxy-4-oxo-2-phenyl-4Hchromen-...)
Affinity DataIC50: 35nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310266BDBM50310266(Hexadecyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7...)
Affinity DataIC50: 48nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310275BDBM50310275(N-Tetradecyl 2-(5-hydroxy-4-oxo-2-phenyl-4Hchromen...)
Affinity DataIC50: 316nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310257BDBM50310257(N-Octadecyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen...)
Affinity DataIC50: 464nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310267BDBM50310267(Octadecyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7...)
Affinity DataIC50: 692nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310265BDBM50310265(Tetradecyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-...)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310274BDBM50310274(N-Dodecyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7...)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310258BDBM50310258(N-Icosyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-...)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310268BDBM50310268(Icosyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-yl...)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310264BDBM50310264(Dodecyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-y...)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310273BDBM50310273(N-Decyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-y...)
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310263BDBM50310263(Decyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-ylo...)
Affinity DataIC50: 3.11E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310272BDBM50310272(N-Nonyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-y...)
Affinity DataIC50: 3.58E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310262BDBM50310262(Nonyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-ylo...)
Affinity DataIC50: 4.96E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310271BDBM50310271(N-Octyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-y...)
Affinity DataIC50: 5.33E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310261BDBM50310261(Octyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-ylo...)
Affinity DataIC50: 5.84E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310270BDBM50310270(N-Heptyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-...)
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310260BDBM50310260(Heptyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-yl...)
Affinity DataIC50: 7.23E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310269BDBM50310269(N-Hexyl-2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-y...)
Affinity DataIC50: 8.71E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Nanjing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50310259BDBM50310259(Hexyl 2-(5-hydroxy-4-oxo-2-phenyl-4H-chromen-7-ylo...)
Affinity DataIC50: 9.12E+3nMAssay Description:Inhibition of EGFR expressed in Sf9 cells assessed as inhibition of receptor autophosphorylation by DELFIA time resolved fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed