Compile Data Set for Download or QSAR
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Found 14 Enz. Inhib. hit(s) with all data for entry = 50031274
TargetMu-type opioid receptor(GUINEA PIG)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310297((2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a,7-...)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310292(CHEMBL604522 | KNT-5)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310294((2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a1-e...)
Affinity DataKi:  26.3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310296((2R,2aS,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Affinity DataKi:  26.4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310297((2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a,7-...)
Affinity DataKi:  193nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310296((2R,2aS,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310294((2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a1-e...)
Affinity DataKi:  275nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310298((2aS,2a1S,5aR)-2a1-(2-(1H-1,2,3-triazol-1-yl)ethyl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310298((2aS,2a1S,5aR)-2a1-(2-(1H-1,2,3-triazol-1-yl)ethyl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310295((2R,2aS,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310293((41R,12R,12aS)-12-((cyclopropylmethyl)(methyl)amin...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310293((41R,12R,12aS)-12-((cyclopropylmethyl)(methyl)amin...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310292(CHEMBL604522 | KNT-5)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50310295((2R,2aS,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed