Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50031281
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50310361(3-(2',6'-Difluorophenyl)-1H-naphtho[2,1-b]pyran-1-...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50310362(3-(2'-Methoxyphenyl)-1H-naphtho[2,1-b]pyran-1-one ...)
Affinity DataEC50:  270nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50310360(3-(2'-Fluorophenyl)-1H-naphtho[2,1-b]pyran-1-one |...)
Affinity DataEC50:  330nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50310363(3-(2'-Pyridinyl)-1H-naphtho[2,1-b]pyran-1-one | CH...)
Affinity DataEC50:  450nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50028963(beta-naphthoflavone | 3-phenyl-1H-benzo[f]chromen-...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50310357(indigo | CHEMBL599552)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50137506(benzo[pqr]tetraphene | benzo[a]pyrene | (B(a)P) | ...)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50310359(3-(2',6'-Dimethylphenyl)-1H-naphtho[2,1-b]pyran-1-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50310358(3-(2'-Methylphenyl)-1H-naphtho[2,1-b]pyran-1-one |...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at aryl hydrocarbon receptor in human MCF7 cells after 24 hrs CYP1A1-dependent EROD assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed