Compile Data Set for Download or QSAR
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Found 28 Enz. Inhib. hit(s) with all data for entry = 50031174
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308527(10-methoxy-N(1)-methylburnamine-17-O-veratrate | C...)
Affinity DataIC50:  500nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308533(CHEMBL589254 | Methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308529(CHEMBL589220 | Methyl (14E)-19-[(benzoyloxy)methyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308528(Alstiphyllanine D | CHEMBL540945)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308532((14E)-14-ethylidene-6-methoxy-19-(methoxycarbonyl)...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308527(10-methoxy-N(1)-methylburnamine-17-O-veratrate | C...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308528(Alstiphyllanine D | CHEMBL540945)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308533(CHEMBL589254 | Methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308531((14E)-19-{[(3,4-dimethoxyphenyl)carbonyloxy]methyl...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308530(CHEMBL602442 | Methyl (14E)-14-ethylidene-6-hydrox...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308532((14E)-14-ethylidene-6-methoxy-19-(methoxycarbonyl)...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308535(CHEMBL601712 | methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308529(CHEMBL589220 | Methyl (14E)-19-[(benzoyloxy)methyl...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308531((14E)-19-{[(3,4-dimethoxyphenyl)carbonyloxy]methyl...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308526(Burnamine-17-O-3',4',5'-trimethoxybenzoate | CHEMB...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308525(Alstiphyllanine F | CHEMBL592521)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308525(Alstiphyllanine F | CHEMBL592521)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308524(Alstiphyllanine E | CHEMBL592477)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308524(Alstiphyllanine E | CHEMBL592477)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308530(CHEMBL602442 | Methyl (14E)-14-ethylidene-6-hydrox...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308526(Burnamine-17-O-3',4',5'-trimethoxybenzoate | CHEMB...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308534(CHEMBL590530 | methyl (14E)-19-[(acetyloxy)methyl]...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308535(CHEMBL601712 | methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  9.70E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308534(CHEMBL590530 | methyl (14E)-19-[(acetyloxy)methyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM20875(1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihyd...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308536(CHEMBL590772 | methyl (14E)-19-[(benzyloxy)methyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308536(CHEMBL590772 | methyl (14E)-19-[(benzyloxy)methyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM20875(1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihyd...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed