Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50039123
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50151001(CHEMBL410478 | (S)-2-((Z)-1-Methyl-3-oxo-3-phenyl-...)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50151001(CHEMBL410478 | (S)-2-((Z)-1-Methyl-3-oxo-3-phenyl-...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315312((S)-2-(4-(2-fluorophenylsulfonyl)piperazin-1-yl)-3...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315312((S)-2-(4-(2-fluorophenylsulfonyl)piperazin-1-yl)-3...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315306((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Affinity DataEC50:  1.14E+3nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315313((S)-2-(4-(4-fluorophenylsulfonyl)piperazin-1-yl)-3...)
Affinity DataEC50:  1.35E+3nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315311((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315311((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Affinity DataEC50:  2.16E+3nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315313((S)-2-(4-(4-fluorophenylsulfonyl)piperazin-1-yl)-3...)
Affinity DataEC50:  2.81E+3nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315306((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Affinity DataEC50:  8.98E+3nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315307((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Affinity DataEC50:  1.06E+4nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  1.06E+4nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315307((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Affinity DataEC50:  1.11E+4nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315309((S)-2-(4-(3-chlorophenyl)piperazin-1-yl)-3-(4-(2-(...)
Affinity DataEC50:  4.52E+4nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315308((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Affinity DataEC50:  5.02E+4nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315308((S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)p...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315309((S)-2-(4-(3-chlorophenyl)piperazin-1-yl)-3-(4-(2-(...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315310((S)-3-(3-bromo-4-(2-(5-methyl-2-phenyloxazol-4-yl)...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GAL4-tagged PPARalpha chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50315310((S)-3-(3-bromo-4-(2-(5-methyl-2-phenyloxazol-4-yl)...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GAL4-tagged PPARgamma chimeric receptor expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2012
Entry Details Article
PubMed