TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Binding affinity to 5HT4 receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Binding affinity to human ERG expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Binding affinity to adrenergic alpha2B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+3nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at alpha4beta2 nAChRMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:Binding affinity to adrenergic alpha2A receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 530nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 390nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 890nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 350nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 1.65E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Agonist activity at rat rat alpha7 nAChR expressed in rat GH4C1 cells by whole cell patch-clamp electrophysiologyMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 260nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech
Curated by ChEMBL
Siena Biotech
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair