Compile Data Set for Download or QSAR
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Found 56 Enz. Inhib. hit(s) with all data for entry = 50039159
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318564((1R,2S,3r,4R,5S,6s)-6-((1-dodecyl-1H-1,2,3-triazol...)
Affinity DataKi:  60nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318563((1R,2S,3r,4R,5S,6s)-6-[(1-Tetradecyl-1H-1,2,3-tria...)
Affinity DataKi:  80nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318562((1R,2S,3r,4R,5S,6s)-6-[(1-Decyl-1H-1,2,3-triazol-4...)
Affinity DataKi:  90nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM18358((2R,3R,4R,5S)-2-(hydroxymethyl)-1-nonylpiperidine-...)
Affinity DataKi:  300nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318560(CHEMBL1083795 | N-decylaminocyclitol)
Affinity DataKi:  300nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318561((1R,2S,3r,4R,5S,6s)-6-[(1-Nonyl-1H-1,2,3-triazol-4...)
Affinity DataKi:  330nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318559((1R,2S,3r,4R,5S,6s)-6-[(1-Octyl-1H-1,2,3-triazol-4...)
Affinity DataKi:  1.80E+3nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318558((1R,2S,3r,4R,5S,6s)-6-((1-(6-propoxyhexyl)-1H-1,2,...)
Affinity DataKi:  2.40E+3nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318557((1R,2S,3r,4R,5S,6s)-6-(3-(1-decyl-1H-1,2,3-triazol...)
Affinity DataKi:  7.60E+3nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318556((1R,2S,3r,4R,5S,6s)-6-[(1-Phenethyl-1H-1,2,3-triaz...)
Affinity DataKi:  1.91E+4nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318554((1R,2S,3r,4R,5S,6s)-6-(3-(1-octyl-1H-1,2,3-triazol...)
Affinity DataKi:  1.99E+4nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318555((1R,2S,3r,4R,5S,6s)-6-[2-(1-Undecyl-1H-1,2,3-triaz...)
Affinity DataKi:  2.02E+4nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318564((1R,2S,3r,4R,5S,6s)-6-((1-dodecyl-1H-1,2,3-triazol...)
Affinity DataIC50:  30nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318564((1R,2S,3r,4R,5S,6s)-6-((1-dodecyl-1H-1,2,3-triazol...)
Affinity DataIC50:  30.2nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318564((1R,2S,3r,4R,5S,6s)-6-((1-dodecyl-1H-1,2,3-triazol...)
Affinity DataIC50:  60nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318563((1R,2S,3r,4R,5S,6s)-6-[(1-Tetradecyl-1H-1,2,3-tria...)
Affinity DataIC50:  89.1nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318562((1R,2S,3r,4R,5S,6s)-6-[(1-Decyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  90nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318563((1R,2S,3r,4R,5S,6s)-6-[(1-Tetradecyl-1H-1,2,3-tria...)
Affinity DataIC50:  90nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318562((1R,2S,3r,4R,5S,6s)-6-[(1-Decyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  93.3nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318562((1R,2S,3r,4R,5S,6s)-6-[(1-Decyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  100nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318563((1R,2S,3r,4R,5S,6s)-6-[(1-Tetradecyl-1H-1,2,3-tria...)
Affinity DataIC50:  100nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318561((1R,2S,3r,4R,5S,6s)-6-[(1-Nonyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  200nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318561((1R,2S,3r,4R,5S,6s)-6-[(1-Nonyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  200nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318561((1R,2S,3r,4R,5S,6s)-6-[(1-Nonyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  224nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM18358((2R,3R,4R,5S)-2-(hydroxymethyl)-1-nonylpiperidine-...)
Affinity DataIC50:  300nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM18358((2R,3R,4R,5S)-2-(hydroxymethyl)-1-nonylpiperidine-...)
Affinity DataIC50:  660nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318559((1R,2S,3r,4R,5S,6s)-6-[(1-Octyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  1.00E+3nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318559((1R,2S,3r,4R,5S,6s)-6-[(1-Octyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318559((1R,2S,3r,4R,5S,6s)-6-[(1-Octyl-1H-1,2,3-triazol-4...)
Affinity DataIC50:  1.10E+3nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318557((1R,2S,3r,4R,5S,6s)-6-(3-(1-decyl-1H-1,2,3-triazol...)
Affinity DataIC50:  1.20E+3nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318560(CHEMBL1083795 | N-decylaminocyclitol)
Affinity DataIC50:  1.80E+3nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318557((1R,2S,3r,4R,5S,6s)-6-(3-(1-decyl-1H-1,2,3-triazol...)
Affinity DataIC50:  3.47E+3nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318557((1R,2S,3r,4R,5S,6s)-6-(3-(1-decyl-1H-1,2,3-triazol...)
Affinity DataIC50:  3.50E+3nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318555((1R,2S,3r,4R,5S,6s)-6-[2-(1-Undecyl-1H-1,2,3-triaz...)
Affinity DataIC50:  4.90E+3nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318558((1R,2S,3r,4R,5S,6s)-6-((1-(6-propoxyhexyl)-1H-1,2,...)
Affinity DataIC50:  6.20E+3nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318558((1R,2S,3r,4R,5S,6s)-6-((1-(6-propoxyhexyl)-1H-1,2,...)
Affinity DataIC50:  7.40E+3nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318556((1R,2S,3r,4R,5S,6s)-6-[(1-Phenethyl-1H-1,2,3-triaz...)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318556((1R,2S,3r,4R,5S,6s)-6-[(1-Phenethyl-1H-1,2,3-triaz...)
Affinity DataIC50:  1.08E+4nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318553((1R,2S,3r,4R,5S,6s)-6-[2-(1-Nonyl-1H-1,2,3-triazol...)
Affinity DataIC50:  1.10E+4nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318558((1R,2S,3r,4R,5S,6s)-6-((1-(6-propoxyhexyl)-1H-1,2,...)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318554((1R,2S,3r,4R,5S,6s)-6-(3-(1-octyl-1H-1,2,3-triazol...)
Affinity DataIC50:  1.82E+4nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318556((1R,2S,3r,4R,5S,6s)-6-[(1-Phenethyl-1H-1,2,3-triaz...)
Affinity DataIC50:  2.50E+4nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318555((1R,2S,3r,4R,5S,6s)-6-[2-(1-Undecyl-1H-1,2,3-triaz...)
Affinity DataIC50:  2.54E+4nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318555((1R,2S,3r,4R,5S,6s)-6-[2-(1-Undecyl-1H-1,2,3-triaz...)
Affinity DataIC50:  2.57E+4nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318554((1R,2S,3r,4R,5S,6s)-6-(3-(1-octyl-1H-1,2,3-triazol...)
Affinity DataIC50:  3.54E+4nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318554((1R,2S,3r,4R,5S,6s)-6-(3-(1-octyl-1H-1,2,3-triazol...)
Affinity DataIC50:  3.55E+4nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318550((1R,2S,3r,4R,5S,6s)-6-(3-(1-hexyl-1H-1,2,3-triazol...)
Affinity DataIC50:  4.46E+4nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318553((1R,2S,3r,4R,5S,6s)-6-[2-(1-Nonyl-1H-1,2,3-triazol...)
Affinity DataIC50:  4.47E+4nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318553((1R,2S,3r,4R,5S,6s)-6-[2-(1-Nonyl-1H-1,2,3-triazol...)
Affinity DataIC50:  4.47E+4nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50318552((1R,2S,3r,4R,5S,6s)-6-[2-(1-Octyl-1H-1,2,3-triazol...)
Affinity DataIC50:  5.59E+4nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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