Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50039222
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50108306BDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321890BDBM50321890(5,6-dichloro-N-(6-(2-methylpyridin-3-yloxy)pyridin...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321867BDBM50321867(6-iodo-5-methyl-N-(pyridin-3-yl)indoline-1-carboxa...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321871BDBM50321871(6-Chloro-5-iodo-2,3-dihydro-indole-1-carboxylic ac...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321861BDBM50321861(5-Iodo-2,3-dihydro-indole-1-carboxylic acid [6-(2-...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321862BDBM50321862(5-bromo-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-yl...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321868BDBM50321868(6-Bromo-5-methyl-2,3-dihydro-indole-1-carboxylic a...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321891BDBM50321891(6-chloro-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50130068BDBM50130068((S)-2-(6-Fluoro-indol-1-yl)-1-methyl-ethylamine | ...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321879BDBM50321879(2-(5-Bromo-indol-1-yl)-1-methyl-ethylamine | (R,S)...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321881BDBM50321881((R,S)-1-(5-fluoro-1H-indol-1-yl)propan-2-amine | 2...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321869BDBM50321869(6-Chloro-5-methyl-2,3-dihydro-indole-1-carboxylic ...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321889BDBM50321889(6-Chloro-5-fluoro-2,3-dihydro-indole-1-carboxylic ...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321863BDBM50321863(5-Chloro-2,3-dihydro-indole-1-carboxylic acid [6-(...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321880BDBM50321880(2-(5-Chloro-indol-1-yl)-1-methyl-ethylamine | (R,S...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321873BDBM50321873(4-bromo-5-methyl-N-(pyridin-3-yl)indoline-1-carbox...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321875BDBM50321875(5,6-dichloro-N-(pyridin-3-yl)indoline-1-carboxamid...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321870BDBM50321870(5-Chloro-6-methyl-2,3-dihydro-indole-1-carboxylic ...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321872BDBM50321872(4-iodo-5-methyl-N-(pyridin-3-yl)indoline-1-carboxa...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321874BDBM50321874(4,5-Dichloro-2,3-dihydro-indole-1-carboxylic acid ...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321864BDBM50321864(5-Fluoro-2,3-dihydro-indole-1-carboxylic acid [6-(...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321886BDBM50321886((E)-5-[(5,6-Dichloro-1H-indol-3-yl)methylene]-2-im...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321876BDBM50321876(6-Chloro-2,3-dihydro-indole-1-carboxylic acid pyri...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321882BDBM50321882((R,S)-1-(5-methyl-1H-indol-1-yl)propan-2-amine | 1...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321867BDBM50321867(6-iodo-5-methyl-N-(pyridin-3-yl)indoline-1-carboxa...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321868BDBM50321868(6-Bromo-5-methyl-2,3-dihydro-indole-1-carboxylic a...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321877BDBM50321877(5-chloro-N-(pyridin-3-yl)indoline-1-carboxamide | ...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321871BDBM50321871(6-Chloro-5-iodo-2,3-dihydro-indole-1-carboxylic ac...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50108306BDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321865BDBM50321865(2,3-Dihydro-indole-1-carboxylic acid [6-(2-methyl-...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321873BDBM50321873(4-bromo-5-methyl-N-(pyridin-3-yl)indoline-1-carbox...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321879BDBM50321879(2-(5-Bromo-indol-1-yl)-1-methyl-ethylamine | (R,S)...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321881BDBM50321881((R,S)-1-(5-fluoro-1H-indol-1-yl)propan-2-amine | 2...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321869BDBM50321869(6-Chloro-5-methyl-2,3-dihydro-indole-1-carboxylic ...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321887BDBM50321887((E)-5-[(6-Chloro-1H-indol-3yl)methylene]-2-imino-1...)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321883BDBM50321883((E)-3-Ethyl-5-[(6-fluoro-1H-indol-3-yl)methylene]-...)
Affinity DataKi:  173nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321880BDBM50321880(2-(5-Chloro-indol-1-yl)-1-methyl-ethylamine | (R,S...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321888BDBM50321888((E)-5-[(6-Fluoro-1H-indol-3-yl)methylene]-2-imino-...)
Affinity DataKi:  235nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50130068BDBM50130068((S)-2-(6-Fluoro-indol-1-yl)-1-methyl-ethylamine | ...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321890BDBM50321890(5,6-dichloro-N-(6-(2-methylpyridin-3-yloxy)pyridin...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321875BDBM50321875(5,6-dichloro-N-(pyridin-3-yl)indoline-1-carboxamid...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321891BDBM50321891(6-chloro-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321870BDBM50321870(5-Chloro-6-methyl-2,3-dihydro-indole-1-carboxylic ...)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321889BDBM50321889(6-Chloro-5-fluoro-2,3-dihydro-indole-1-carboxylic ...)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321885BDBM50321885((E)-5-((1H-Indol-3yl)methylene)-2-imino-1,3-dimeth...)
Affinity DataKi:  598nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321874BDBM50321874(4,5-Dichloro-2,3-dihydro-indole-1-carboxylic acid ...)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321884BDBM50321884((Z)-5-((1H-Indol-3yl)methylene)-3-ethyl-2-imino-1-...)
Affinity DataKi:  655nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321866BDBM50321866(6,7-Dichloro-2,3-dihydro-indole-1-carboxylic acid ...)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321882BDBM50321882((R,S)-1-(5-methyl-1H-indol-1-yl)propan-2-amine | 1...)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of North Texas Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321876BDBM50321876(6-Chloro-2,3-dihydro-indole-1-carboxylic acid pyri...)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
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