Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50004366
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482233BDBM50482233(CHEMBL1163161)
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482232BDBM50482232(CHEMBL1165020)
Affinity DataIC50: 80nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 19149BDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482238BDBM50482238(CHEMBL1164069)
Affinity DataIC50: 250nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478021BDBM50478021(CHEMBL402341)
Affinity DataIC50: 450nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482239BDBM50482239(CHEMBL1163989)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482243BDBM50482243(CHEMBL1163582)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482235BDBM50482235(CHEMBL1165800)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482242BDBM50482242(ACS 5)
Affinity DataIC50: 4.64E+4nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482241BDBM50482241(CHEMBL1163626)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482237BDBM50482237(CHEMBL1163984)
Affinity DataIC50: 8.29E+4nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482236BDBM50482236(CHEMBL1163983)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482234BDBM50482234(CHEMBL1163627)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482240BDBM50482240(CHEMBL1163674)
Affinity DataIC50: 1.79E+5nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sulfidris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50482244BDBM50482244(CHEMBL1163624)
Affinity DataIC50: 9.19E+5nMAssay Description:Inhibition of HDAC in human HeLa cells extracts after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed