Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50032512
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034839(Ro-15-1310 | 8-Chloro-5-methyl-6-oxo-5,6-dihydro-4...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to human recombinant GABA alpha-1-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034839(Ro-15-1310 | 8-Chloro-5-methyl-6-oxo-5,6-dihydro-4...)
Affinity DataKi:  9.20nMAssay Description:Binding affinity to human recombinant GABA alpha-3-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034839(Ro-15-1310 | 8-Chloro-5-methyl-6-oxo-5,6-dihydro-4...)
Affinity DataKi:  16.3nMAssay Description:Binding affinity to human recombinant GABA alpha-2-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGABA A receptor alpha-4/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi:  38.8nMAssay Description:Binding affinity to human recombinant GABA alpha-4-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha-5-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha-1-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha-2-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha-3-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGABA A receptor alpha-4/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  2.61E+3nMAssay Description:Binding affinity to human recombinant GABA alpha-4-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  1.75E+4nMAssay Description:Binding affinity to human recombinant GABA alpha-1-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  2.21E+4nMAssay Description:Binding affinity to human recombinant GABA alpha-3-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  2.95E+4nMAssay Description:Binding affinity to human recombinant GABA alpha-5-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Human)
University of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  3.38E+4nMAssay Description:Binding affinity to human recombinant GABA alpha-2-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed