Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50032180
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325605((R)-methyl 8-(3-(4-(2,2-diphenylacetamido)-5-(4-hy...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50060728((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325608((R)-1-[4-(2,2-Diphenylacetamido)-5-(4-hydroxybenzy...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325609((R)-2-{4-[4-(Ammoniomethyl)-1H-1,2,3-triazol-1-yl]...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325604((R)-benzyl 4-(2,2-diphenylacetamido)-1-(4-hydroxyp...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325610((13R)-13-(4-Hydroxybenzylcarbamoyl)-3,6,15-trioxo-...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325613((R)-18-Amino-4-(2,2-diphenylacetamido)-1-(4-hydrox...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325603(CHEMBL1223990 | N-((R)-4-(2,2-diphenylacetamido)-1...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325611((R)-21-Carboxy-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325606((4R,12R,13S,14R,15R)-12,13,14,15-Tetraacetoxy-4-(2...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325612((R)-4-(2,2-Diphenylacetamido)-1-(4-hydroxyphenyl)-...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325607((R)-21-(4-Hydroxybenzylcarbamoyl)-3,7,14,23-tetrao...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325602((R)-2-(2,2-diphenylacetamido)-N-(4-hydroxybenzyl)-...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325601((R)-N-(N-(4-(2,2-diphenylacetamido)-5-(4-hydroxybe...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50325600((R)-N-(N-(4-(2,2-diphenylacetamido)-5-(4-hydroxybe...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]UR-MK114 from NPY1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed