Compile Data Set for Download or QSAR
maximum 50k data
Found 74 Enz. Inhib. hit(s) with all data for entry = 50041848
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215615(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  1.20nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215583(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215655(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215645(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  1.90nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215579(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  2.10nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215607(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  2.40nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215629(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  2.70nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215578(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  2.80nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215613(3-(2,6-dichloropyridin-4-yl)-1-((3R,6S)-6-(3-((dim...)
Affinity DataKi:  3.30nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215614(3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino...)
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215640(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  4.40nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215650(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  4.5nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215611(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  4.98nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215634(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  5.20nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215610(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  5.40nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215591(3-(3-bromophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicy...)
Affinity DataKi:  5.70nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215609(3-(3-chlorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bic...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215619(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  7nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215641(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  7.19nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215636(3-(3-cyanophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bicy...)
Affinity DataKi:  7.60nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215651(1-((3R,6S)-6-(3-bromophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  7.76nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215624(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  8.71nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215637(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  8.71nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215625(3-(2,6-dichloropyridin-4-yl)-1-((3R,6S)-6-(3-(((S)...)
Affinity DataKi:  8.89nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215586(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  9.40nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215642(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  9.71nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215649(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  10.4nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215652(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  11.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215603(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  11.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215589(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  12.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215594(3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino...)
Affinity DataKi:  13nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215659(1-(4-(2-(aminomethyl)thiazol-5-yl)cyclohex-3-enyl)...)
Affinity DataKi:  13nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50416850(CHEMBL1253196)
Affinity DataKi:  15nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50416852(CHEMBL1254636)
Affinity DataKi:  15nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215658(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-((dime...)
Affinity DataKi:  15nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215590(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  15nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215605(3-(3-chloro-4-fluorophenyl)-1-((3R,6S)-6-(3-cyanop...)
Affinity DataKi:  15nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50416847(CHEMBL1254714)
Affinity DataKi:  15nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50416845(CHEMBL1254564)
Affinity DataKi:  16nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215588(1-(4-(5-(aminomethyl)thiazol-2-yl)cyclohex-3-enyl)...)
Affinity DataKi:  17.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215643(3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino...)
Affinity DataKi:  18.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215635(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  20nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215633(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  20nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215626(3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino...)
Affinity DataKi:  21.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215587(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  21.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50416846(CHEMBL1254713)
Affinity DataKi:  22.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50416849(CHEMBL1254560)
Affinity DataKi:  23.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215606(1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3...)
Affinity DataKi:  26nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215647(3-(3-chlorophenyl)-1-((3R,6S)-6-(3-cyanophenyl)bic...)
Affinity DataKi:  27.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Universidad De Cartagena

Curated by ChEMBL
LigandPNGBDBM50215601(3-(3-chloro-4-fluorophenyl)-1-(2-(diisopropylamino...)
Affinity DataKi:  29.0nMAssay Description:Antagonist activity at MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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