Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50032197
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325847(N-(cyclopropylmethyl)-2-(6-(3-morpholinopropoxy)-4...)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325825((S)-2-amino-N-((S)-1-(3-(2-(cyclopropylmethylamino...)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325847(N-(cyclopropylmethyl)-2-(6-(3-morpholinopropoxy)-4...)
Affinity DataIC50: 210nMAssay Description:Displacement of [3H]AVP from rat vasopressin V3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325842(N-(cyclopropylmethyl)-2-(4-oxo-2-phenyl-6-(3-(pipe...)
Affinity DataIC50: 310nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325844(2-(6-(3-(azepan-1-yl)propoxy)-4-oxo-2-phenylquinaz...)
Affinity DataIC50: 340nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325845(N-(cyclopropylmethyl)-2-(6-(3-(4-methoxypiperidin-...)
Affinity DataIC50: 710nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325846(N-(cyclopropylmethyl)-2-(6-(3-(4-hydroxypiperidin-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325837(N-(cyclopropylmethyl)-2-(6-(3-(4-methylpiperazin-1...)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325843(N-(cyclopropylmethyl)-2-(4-oxo-2-phenyl-6-(3-(pyrr...)
Affinity DataIC50: 1.80E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325830((S)-2-(6-(2-amino-4-methylpentyloxy)-4-oxo-2-pheny...)
Affinity DataIC50: 2.10E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325832(2-(6-(3-aminopropoxy)-4-oxo-2-phenylquinazolin-3(4...)
Affinity DataIC50: 3.60E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325841(N-(cyclopropylmethyl)-2-(6-(3-(diethylamino)propox...)
Affinity DataIC50: 3.80E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325831(2-(6-(2-aminoethoxy)-4-oxo-2-phenylquinazolin-3(4H...)
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325838(N-(cyclopropylmethyl)-2-(6-(4-(4-methylpiperazin-1...)
Affinity DataIC50: 4.80E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325826((S)-2-amino-N-(1-(3-(2-(cyclopropylmethylamino)-2-...)
Affinity DataIC50: 5.10E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325840(N-(cyclopropylmethyl)-2-(6-(3-(methylamino)propoxy...)
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325836(N-(cyclopropylmethyl)-2-(6-(2-(4-methylpiperazin-1...)
Affinity DataIC50: 2.20E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325839(N-(cyclopropylmethyl)-2-(4-oxo-2-phenyl-6-(3-(pipe...)
Affinity DataIC50: 2.58E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325834(2-(6-(5-aminopentyloxy)-4-oxo-2-phenylquinazolin-3...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325833(2-(6-(4-aminobutoxy)-4-oxo-2-phenylquinazolin-3(4H...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325827(2-amino-N-(2-(3-(2-(cyclopropylmethylamino)-2-oxoe...)
Affinity DataIC50: 3.05E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325847(N-(cyclopropylmethyl)-2-(6-(3-morpholinopropoxy)-4...)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325835(2-(6-(6-aminohexyloxy)-4-oxo-2-phenylquinazolin-3(...)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325847(N-(cyclopropylmethyl)-2-(6-(3-morpholinopropoxy)-4...)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325828(N-(2-(3-(2-(cyclopropylmethylamino)-2-oxoethyl)-4-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325829(N-(cyclopropylmethyl)-2-(6-hydroxy-4-oxo-2-phenylq...)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed