Compile Data Set for Download or QSAR
maximum 50k data
Found 99 Enz. Inhib. hit(s) with all data for entry = 50032582
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331461(1-Trifluoromethyl-cyclopropanecarboxylic acid{3-[(...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331462(1-Trifluoromethyl-cyclobutanecarboxylic acid{3-[(6...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331463(2,2-Difluoro-cyclopropanecarboxylic acid{3-[(6-flu...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331464(3,3,3-Trifluoro-N-{3-[(6-fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331465(CHEMBL1290510 | Furan-3-carboxylic acid{3-[(6-fluo...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331466(CHEMBL1290169 | N-{3-[(1,1-Dioxo-1H-1lambda*6*-ben...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331467(1-Methyl-cyclopropanecarboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331468(CHEMBL1290509 | Furan-2-carboxylic acid{3-[(6-fluo...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331469(CHEMBL1289300 | N-{3-[(6-Fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331470(CHEMBL1289188 | Pyrazine-2-carboxylic acid{3-[(6-f...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331461(1-Trifluoromethyl-cyclopropanecarboxylic acid{3-[(...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331471(3,3,3-Trifluoro-N-{3-[(6-fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331464(3,3,3-Trifluoro-N-{3-[(6-fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331472(CHEMBL1289068 | Cyclopropanecarboxylic acid{3-[(6-...)
Affinity DataIC50:  280nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331473(CHEMBL1290621 | Thiazole-4-carboxylic acid{3-[(6-f...)
Affinity DataIC50:  290nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331474(CHEMBL1290618 | Pyrrole-1-carboxylic acid{3-[(6-fl...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331475(3-Hydroxy-pyridine-2-carboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331462(1-Trifluoromethyl-cyclobutanecarboxylic acid{3-[(6...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331463(2,2-Difluoro-cyclopropanecarboxylic acid{3-[(6-flu...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331476(4-Cyano-tetrahydro-pyran-4-carboxylic acid{3-[(6-f...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331477(CHEMBL1290280 | Morpholine-4-carboxylic acid{3-[(6...)
Affinity DataIC50:  340nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331474(CHEMBL1290618 | Pyrrole-1-carboxylic acid{3-[(6-fl...)
Affinity DataIC50:  340nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331479(1-Hydroxy-cyclohexanecarboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331478(1-Cyano-cyclopropanecarboxylic acid{3-[(6-fluoro-1...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331470(CHEMBL1289188 | Pyrazine-2-carboxylic acid{3-[(6-f...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331480(CHEMBL1289744 | Tetrahydro-furan-2-carboxylic acid...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331465(CHEMBL1290510 | Furan-3-carboxylic acid{3-[(6-fluo...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331467(1-Methyl-cyclopropanecarboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331469(CHEMBL1289300 | N-{3-[(6-Fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331481(4,4-Difluoro-1-hydroxy-cyclohexanecarboxylic acid{...)
Affinity DataIC50:  390nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331468(CHEMBL1290509 | Furan-2-carboxylic acid{3-[(6-fluo...)
Affinity DataIC50:  410nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331482(CHEMBL1290170 | N-{3-[(1,1-Dioxo-1H-1lambda*6*-ben...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331483(CHEMBL1289850 | Tetrahydro-pyran-2-carboxylic acid...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331479(1-Hydroxy-cyclohexanecarboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50:  450nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331475(3-Hydroxy-pyridine-2-carboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50:  460nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331484(1-Hydroxy-cyclopentanecarboxylic acid{3-[(6-fluoro...)
Affinity DataIC50:  470nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331485(CHEMBL1290279 | Morpholine-4-carboxylic acid{3-[(1...)
Affinity DataIC50:  470nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331471(3,3,3-Trifluoro-N-{3-[(6-fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50:  480nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331472(CHEMBL1289068 | Cyclopropanecarboxylic acid{3-[(6-...)
Affinity DataIC50:  490nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331486(1-Methyl-1H-imidazole-2-carboxylic acid{3-[(6-fluo...)
Affinity DataIC50:  520nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331487(1-Amino-cyclopropanecarboxylic acid{3-[(6-fluoro-1...)
Affinity DataIC50:  530nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331488(CHEMBL1290508 | Tetrahydro-pyran-4-carboxylic acid...)
Affinity DataIC50:  530nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331473(CHEMBL1290621 | Thiazole-4-carboxylic acid{3-[(6-f...)
Affinity DataIC50:  540nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331478(1-Cyano-cyclopropanecarboxylic acid{3-[(6-fluoro-1...)
Affinity DataIC50:  540nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331423(CHEMBL1289183 | N-{3-[(1,1-Dioxo-1H-1lambda*6*-ben...)
Affinity DataIC50:  550nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331486(1-Methyl-1H-imidazole-2-carboxylic acid{3-[(6-fluo...)
Affinity DataIC50:  550nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331489(CHEMBL1290395 | N-{3-[(1,1-Dioxo-1H-1lambda*6*-ben...)
Affinity DataIC50:  560nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331476(4-Cyano-tetrahydro-pyran-4-carboxylic acid{3-[(6-f...)
Affinity DataIC50:  560nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331481(4,4-Difluoro-1-hydroxy-cyclohexanecarboxylic acid{...)
Affinity DataIC50:  630nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331483(CHEMBL1289850 | Tetrahydro-pyran-2-carboxylic acid...)
Affinity DataIC50:  640nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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