Compile Data Set for Download or QSAR
maximum 50k data
Found 69 Enz. Inhib. hit(s) with all data for entry = 50032792
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334828(CHEMBL1643160 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334828(CHEMBL1643160 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334829(CHEMBL1643161 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334829(CHEMBL1643161 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334825(2-(4-(3-chlorophenyl)piperazin-1-yl)-N-(4-(5-cyano...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334825(2-(4-(3-chlorophenyl)piperazin-1-yl)-N-(4-(5-cyano...)
Affinity DataIC50:  29nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334815(2-(1-(benzylsulfonyl)piperidin-4-yloxy)-N-(4-(5-cy...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334832(CHEMBL1643164 | ethyl 4-(4-(2-(4-(5-cyano-7-methyl...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334820(CHEMBL1643153 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  49nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334830(CHEMBL1643162 | methyl 3-(4-(2-(4-(5-cyano-7-methy...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334826(2-(4-(4-chlorophenyl)piperazin-1-yl)-N-(4-(5-cyano...)
Affinity DataIC50:  53nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334822(CHEMBL1641618 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334832(CHEMBL1643164 | ethyl 4-(4-(2-(4-(5-cyano-7-methyl...)
Affinity DataIC50:  59nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334830(CHEMBL1643162 | methyl 3-(4-(2-(4-(5-cyano-7-methy...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334818(CHEMBL1642947 | tert-butyl 4-(2-(4-(5-cyano-7-meth...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334827(CHEMBL1643159 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  65nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334824(2-(4-(2-chlorophenyl)piperazin-1-yl)-N-(4-(5-cyano...)
Affinity DataIC50:  69nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334796(CHEMBL1642925 | N-(4-(5-cyanobenzo[d]oxazol-2-yl)p...)
Affinity DataIC50:  72nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334809(CHEMBL1642938 | tert-butyl 2-(4-(2-(4-(5-cyano-7-m...)
Affinity DataIC50:  83nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334818(CHEMBL1642947 | tert-butyl 4-(2-(4-(5-cyano-7-meth...)
Affinity DataIC50:  83nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334806(CHEMBL1642935 | tert-pentyl 4-(2-(4-(5-cyano-7-met...)
Affinity DataIC50:  84nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334801(CHEMBL1642930 | tert-butyl 4-(2-(4-(5-cyano-7-meth...)
Affinity DataIC50:  91nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334801(CHEMBL1642930 | tert-butyl 4-(2-(4-(5-cyano-7-meth...)
Affinity DataIC50:  92nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334795(CHEMBL1642924 | N-(4-(5-cyanobenzo[d]oxazol-2-yl)p...)
Affinity DataIC50:  92nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334806(CHEMBL1642935 | tert-pentyl 4-(2-(4-(5-cyano-7-met...)
Affinity DataIC50:  94nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334804(CHEMBL1642933 | isopropyl 4-(2-(4-(5-cyano-7-methy...)
Affinity DataIC50:  99nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334823(CHEMBL1643155 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  99nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334823(CHEMBL1643155 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  109nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334821(CHEMBL1643154 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  111nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334805(CHEMBL1642934 | neopentyl 4-(2-(4-(5-cyano-7-methy...)
Affinity DataIC50:  111nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334797(CHEMBL1642926 | N-(4-(5-cyanobenzo[d]oxazol-2-yl)p...)
Affinity DataIC50:  115nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334822(CHEMBL1641618 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  123nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334808(CHEMBL1642937 | benzyl 4-(2-(4-(5-cyano-7-methylbe...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334805(CHEMBL1642934 | neopentyl 4-(2-(4-(5-cyano-7-methy...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334826(2-(4-(4-chlorophenyl)piperazin-1-yl)-N-(4-(5-cyano...)
Affinity DataIC50:  135nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334794(CHEMBL1642923 | N-(4-(5-cyanobenzo[d]oxazol-2-yl)p...)
Affinity DataIC50:  146nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334804(CHEMBL1642933 | isopropyl 4-(2-(4-(5-cyano-7-methy...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334815(2-(1-(benzylsulfonyl)piperidin-4-yloxy)-N-(4-(5-cy...)
Affinity DataIC50:  169nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334809(CHEMBL1642938 | tert-butyl 2-(4-(2-(4-(5-cyano-7-m...)
Affinity DataIC50:  181nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334813(2-(1-(butylsulfonyl)piperidin-4-yloxy)-N-(4-(5-cya...)
Affinity DataIC50:  207nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334807(CHEMBL1642936 | phenyl 4-(2-(4-(5-cyano-7-methylbe...)
Affinity DataIC50:  221nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334810(CHEMBL1642939 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  228nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334808(CHEMBL1642937 | benzyl 4-(2-(4-(5-cyano-7-methylbe...)
Affinity DataIC50:  252nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334803(CHEMBL1642932 | ethyl 4-(2-(4-(5-cyano-7-methylben...)
Affinity DataIC50:  254nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334811(CHEMBL1642940 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  256nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334793(CHEMBL1642922 | N-(4-(5-cyanobenzo[d]oxazol-2-yl)p...)
Affinity DataIC50:  280nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334800(CHEMBL1642929 | tert-butyl 4-(2-(4-(5-cyanobenzo[d...)
Affinity DataIC50:  287nMAssay Description:Inhibition of CETP-mediated cholesteryl ester transfer in human serum after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334814(CHEMBL1642943 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  336nMAssay Description:Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334820(CHEMBL1643153 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  349nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334810(CHEMBL1642939 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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