Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50041880
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417614(CHEMBL1645396)
Affinity DataEC50:  2nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417607(CHEMBL1645401)
Affinity DataEC50:  3.98nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417617(CHEMBL1645392)
Affinity DataEC50:  3.98nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417611(CHEMBL1641638)
Affinity DataEC50:  5.01nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417613(CHEMBL1645400)
Affinity DataEC50:  6.31nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417617(CHEMBL1645392)
Affinity DataEC50:  7.94nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417608(CHEMBL1645399)
Affinity DataEC50:  10nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417615(CHEMBL1645402)
Affinity DataEC50:  12.6nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417612(CHEMBL1645395)
Affinity DataEC50:  12.6nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417616(CHEMBL1645403)
Affinity DataEC50:  12.6nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417606(CHEMBL1645398)
Affinity DataEC50:  25.1nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417609(CHEMBL1645397)
Affinity DataEC50:  25.1nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417610(CHEMBL1645394)
Affinity DataEC50:  31.6nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417614(CHEMBL1645396)
Affinity DataEC50:  50.1nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417613(CHEMBL1645400)
Affinity DataEC50:  79.4nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417616(CHEMBL1645403)
Affinity DataEC50:  100nMAssay Description:Antagonist activity at human GR DNA binding domain transfected in CHO cells co-transfected with MMTV-luciferase gene assessed as inhibition of cortis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417612(CHEMBL1645395)
Affinity DataEC50:  126nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417611(CHEMBL1641638)
Affinity DataEC50:  200nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417610(CHEMBL1645394)
Affinity DataEC50:  200nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417609(CHEMBL1645397)
Affinity DataEC50:  251nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417608(CHEMBL1645399)
Affinity DataEC50:  631nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417606(CHEMBL1645398)
Affinity DataEC50:  794nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417607(CHEMBL1645401)
Affinity DataEC50:  794nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417605(CHEMBL1645393)
Affinity DataEC50:  1.00E+3nMAssay Description:Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417616(CHEMBL1645403)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human MR ligand binding domain transfected in CHO cells co-transfected with MMTV-luciferase gene assessed as inhibition of cor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417605(CHEMBL1645393)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417615(CHEMBL1645402)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417616(CHEMBL1645403)
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed