Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50032860
TargetPolyphenol oxidase 2(White button mushroom)
University of California

Curated by ChEMBL
LigandPNGBDBM50236983(2-hydroxycyclohepta-2,4,6-trienone | tropolone | 2...)
Affinity DataIC50: 400nMAssay Description:Inhibition of mushroom tyrosinase after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335802(4-Fluoro-N-(8-hydroxyquinolin-7-yl)benzenesulfonam...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetPolyphenol oxidase 2(White button mushroom)
University of California

Curated by ChEMBL
LigandPNGBDBM50335803(3-hydroxy-2-methyl-4H-pyran-4-thione | CHEMBL16506...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of mushroom tyrosinase after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335813(N-(8-Hydroxyquinolin-7-yl)-[1,1-biphenyl]-4-sulfon...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335814(N-(8-Hydroxyquinolin-7-yl)thiophene-2-sulfonamide ...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335807(N-(8-Hydroxyquinolin-7-yl)benzenesulfonamide | CHE...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335805(4-Fluoro-N-(8-hydroxyquinolin-5-yl)benzenesulfonam...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335812(N-(8-Hydroxyquinolin-5-yl)thiophene-2-sulfonamide ...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335804(N-(8-Hydroxyquinolin-5-yl)benzenesulfonamide | CHE...)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335801(N-(8-Hydroxyquinolin-5-yl)-[1,1'-biphenyl]-4-sulfo...)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335803(3-hydroxy-2-methyl-4H-pyran-4-thione | CHEMBL16506...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human recombinant 5-lipoxygenase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335808(2,5-Dihydroxybenzoate, VI | gentisic acid | CHEMBL...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of human recombinant 5-lipoxygenase after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335806(3-hydroxy-4H-pyran-4-thione | CHEMBL1649594)
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetPolyphenol oxidase 2(White button mushroom)
University of California

Curated by ChEMBL
LigandPNGBDBM26193(salicylic acid | 2-Hydroxybenzoate, I | CHEMBL424 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mushroom tyrosinase after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335810(2-thiouracil | 4-mercaptopyrimidin-2-ol | CHEMBL16...)
Affinity DataIC50: 1.21E+5nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM32203(cid_1923 | CHEMBL310555 | 8-quinolinol | quinolin-...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50236983(2-hydroxycyclohepta-2,4,6-trienone | tropolone | 2...)
Affinity DataIC50: 1.46E+5nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetPolyphenol oxidase 2(White button mushroom)
University of California

Curated by ChEMBL
LigandPNGBDBM50335809(6-hydroxypicolinic acid | CHEMBL1650602)
Affinity DataIC50: 1.59E+5nMAssay Description:Inhibition of mushroom tyrosinase after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLethal factor(Bacillus anthracis)
University of California

Curated by ChEMBL
LigandPNGBDBM50335806(3-hydroxy-4H-pyran-4-thione | CHEMBL1649594)
Affinity DataIC50: 2.04E+5nMAssay Description:Inhibition of recombinant anthrax lethal factor after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50335811(3-amino-2-hydroxybenzoic acid | CHEMBL1650630)
Affinity DataIC50: 3.89E+5nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLethal factor(Bacillus anthracis)
University of California

Curated by ChEMBL
LigandPNGBDBM50099857(acetohydroxamic acid | AHA | Acethydroxamsaeure | ...)
Affinity DataIC50: 1.14E+7nMAssay Description:Inhibition of recombinant anthrax lethal factor after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50099857(acetohydroxamic acid | AHA | Acethydroxamsaeure | ...)
Affinity DataIC50: 1.50E+7nMAssay Description:Inhibition of human recombinant MMP2 after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed