Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50032711
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333579BDBM50333579(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)q...)
Affinity DataIC50: 140nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333582BDBM50333582(6-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)-...)
Affinity DataIC50: 300nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333581BDBM50333581(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)-...)
Affinity DataIC50: 310nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333586BDBM50333586(2-{2-[3-Methoxy-4-(4-methyl-imidazol-1-yl)-phenyl]...)
Affinity DataIC50: 390nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333584BDBM50333584(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)b...)
Affinity DataIC50: 510nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333587BDBM50333587(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)-...)
Affinity DataIC50: 680nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333593BDBM50333593(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)-...)
Affinity DataIC50: 870nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333583BDBM50333583(ethyl 4-amino-2-(3-methoxy-4-(4-methyl-1H-imidazol...)
Affinity DataIC50: 980nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333580BDBM50333580(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)-...)
Affinity DataIC50: 990nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333585BDBM50333585(Benzyl-(2-{2-[3-methoxy-4-(4-methyl-imidazol-1-yl)...)
Affinity DataIC50: 1.12E+3nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333578BDBM50333578(2-{(E)-2-[3-Methoxy-4-(4-methyl-imidazol-1-yl)-phe...)
Affinity DataIC50: 4.73E+3nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333590BDBM50333590(7-chloro-2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333591BDBM50333591(7-bromo-2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333592BDBM50333592(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333576BDBM50333576(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333577BDBM50333577(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333588BDBM50333588(2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)styryl)q...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333589BDBM50333589(6-fluoro-2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of radiolabeled MK-499 from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed