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Found 52 Enz. Inhib. hit(s) with all data for entry = 50039379
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336806(1-(3-(aminomethyl)-2-isobutyl-4-p-tolylquinolin-6-...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336818(5-(Aminomethyl)-2-benzyl-6-(2,2-dimethylpropyl)-4-...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336815(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336817(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336820(CHEMBL1672127 | [5-(Aminomethyl)-6-(2,2-dimethylpr...)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336814(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-(...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336805(6-[3-(Aminomethyl)-4-(4-methylphenyl)-2-(2-methylp...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336803(4-[3-(Aminomethyl)-4-(4-methylphenyl)-2-(2-methylp...)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336804(5-[3-(Aminomethyl)-4-(4-methylphenyl)-2-(2-methylp...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336819(CHEMBL1672126 | [5-(Aminomethyl)-6-(2,2-dimethylpr...)
Affinity DataIC50:  10nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336813(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50333184(5-(aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-m...)
Affinity DataIC50:  18nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336816(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-(1-methyl...)
Affinity DataIC50:  19nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336808(CHEMBL1672115 | [5-(Aminomethyl)-2-methyl-4-(4-met...)
Affinity DataIC50:  20nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336802(3-[3-(Aminomethyl)-4-(4-methylphenyl)-2-(2-methylp...)
Affinity DataIC50:  23nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336809(3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(...)
Affinity DataIC50:  39nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336811(5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-prop...)
Affinity DataIC50:  57nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336812(5-(Aminomethyl)-6-butyl-2-methyl-4-(4-methylphenyl...)
Affinity DataIC50:  58nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336810((2E)-3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl...)
Affinity DataIC50:  66nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336818(5-(Aminomethyl)-2-benzyl-6-(2,2-dimethylpropyl)-4-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336817(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50:  420nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336815(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50:  630nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336814(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-(...)
Affinity DataIC50:  820nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336809(3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336817(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336816(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-(1-methyl...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336815(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336815(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336818(5-(Aminomethyl)-2-benzyl-6-(2,2-dimethylpropyl)-4-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336816(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-(1-methyl...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336814(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-(...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336817(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336814(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-(...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50333184(5-(aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-m...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336818(5-(Aminomethyl)-2-benzyl-6-(2,2-dimethylpropyl)-4-...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336813(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336812(5-(Aminomethyl)-6-butyl-2-methyl-4-(4-methylphenyl...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50333184(5-(aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-m...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336816(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-(1-methyl...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336813(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336813(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336808(CHEMBL1672115 | [5-(Aminomethyl)-2-methyl-4-(4-met...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336809(3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336808(CHEMBL1672115 | [5-(Aminomethyl)-2-methyl-4-(4-met...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50333184(5-(aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-m...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336809(3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Rattus norvegicus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336808(CHEMBL1672115 | [5-(Aminomethyl)-2-methyl-4-(4-met...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336820(CHEMBL1672127 | [5-(Aminomethyl)-6-(2,2-dimethylpr...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336819(CHEMBL1672126 | [5-(Aminomethyl)-6-(2,2-dimethylpr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336820(CHEMBL1672127 | [5-(Aminomethyl)-6-(2,2-dimethylpr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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