Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50032937
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336669(N-[(6beta,14beta-Epoxy-3-hydroxy-17-methylmorphina...)
Affinity DataKi:  0.0522nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336672(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.0754nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336674(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.0812nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336664((2E)-N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3...)
Affinity DataKi:  0.0828nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336677(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.0833nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336673(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.0880nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336670(N-[(6beta,14beta-Epoxy-3-hydroxy-17-isobutylmorphi...)
Affinity DataKi:  0.108nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336667(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.109nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336674(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336679(N-[(6beta,14beta-Epoxy-3-hydroxy-17-isobutylmorphi...)
Affinity DataKi:  0.116nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336667(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336671(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336672(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.121nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336663(2-Phenyl-N-[(17-cyclopropylmethyl-6beta,14beta-epo...)
Affinity DataKi:  0.124nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336666(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336665(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.129nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336665(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.132nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336663(2-Phenyl-N-[(17-cyclopropylmethyl-6beta,14beta-epo...)
Affinity DataKi:  0.132nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336683(N-[(17-Cyclobutylmethyl-6beta,14beta-epoxy-3-hydro...)
Affinity DataKi:  0.133nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336661(N-{[(1R,9R,10S,13S)-17-(cyclopropylmethyl)-4-hydro...)
Affinity DataKi:  0.134nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336661(N-{[(1R,9R,10S,13S)-17-(cyclopropylmethyl)-4-hydro...)
Affinity DataKi:  0.135nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336683(N-[(17-Cyclobutylmethyl-6beta,14beta-epoxy-3-hydro...)
Affinity DataKi:  0.138nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336680(N-[(6beta,14beta-Epoxy-3-hydroxy-17-isobutylmorphi...)
Affinity DataKi:  0.141nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336673(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.147nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336664((2E)-N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3...)
Affinity DataKi:  0.147nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336666(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.156nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336677(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.182nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336662(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.188nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50325534(nalfurafine | CHEMBL267495)
Affinity DataKi:  0.225nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336669(N-[(6beta,14beta-Epoxy-3-hydroxy-17-methylmorphina...)
Affinity DataKi:  0.228nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336676(N-[(6beta,14beta-Epoxy-3-hydroxy-17-phenethylmorph...)
Affinity DataKi:  0.243nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336668(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336670(N-[(6beta,14beta-Epoxy-3-hydroxy-17-isobutylmorphi...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336662(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.326nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336671(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.384nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336679(N-[(6beta,14beta-Epoxy-3-hydroxy-17-isobutylmorphi...)
Affinity DataKi:  0.389nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336687(N-[(17-Benzyl-6beta,14beta-epoxy-3-hydroxymorphina...)
Affinity DataKi:  0.438nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336680(N-[(6beta,14beta-Epoxy-3-hydroxy-17-isobutylmorphi...)
Affinity DataKi:  0.466nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336681(N-[(17-benzyl-6beta,14beta-epoxy-3-hydroxymorphina...)
Affinity DataKi:  0.543nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50325534(nalfurafine | CHEMBL267495)
Affinity DataKi:  0.582nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336685(N-[(17-Benzyl-6beta,14beta-epoxy-3-hydroxymorphina...)
Affinity DataKi:  0.699nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336668(N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydr...)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NORBNI | NOR-BNI (HCI)2)
Affinity DataKi:  0.861nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336678(N-[(6beta,14beta-Epoxy-3-hydroxy-17-isobutylmorphi...)
Affinity DataKi:  0.946nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336675(N-[(17-Benzyl-6beta,14beta-epoxy-3-hydroxymorphina...)
Affinity DataKi:  1.05nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336676(N-[(6beta,14beta-Epoxy-3-hydroxy-17-phenethylmorph...)
Affinity DataKi:  1.12nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336684(N-[(17-Benzyl-6beta,14beta-epoxy-3-hydroxymorphina...)
Affinity DataKi:  1.13nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336687(N-[(17-Benzyl-6beta,14beta-epoxy-3-hydroxymorphina...)
Affinity DataKi:  1.35nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336682(N-[(17-Benzyl-6beta,14beta-epoxy-3-hydroxymorphina...)
Affinity DataKi:  1.82nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50336678(N-[(6beta,14beta-Epoxy-3-hydroxy-17-isobutylmorphi...)
Affinity DataKi:  2.31nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
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