Compile Data Set for Download or QSAR
Report error Found 375 Enz. Inhib. hit(s) with all data for entry = 50033028
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 11162BDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338432BDBM50338432((R)-1-(1-(5-(aminooxycarbonyl)pyridin-3-yl)piperid...)
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338439BDBM50338439(3-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethyl)pipe...)
Affinity DataIC50: 21nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140533BDBM50140533(N-[4-((S)-1-Amino-2-oxo-2-thiazolidin-3-yl-ethyl)-...)
Affinity DataIC50: 22nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338440BDBM50338440(trans-N-(4-((S)-1-amino-2-oxo-2-(thiazolidin-3-yl)...)
Affinity DataIC50: 33nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338458BDBM50338458(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 38nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338438BDBM50338438(3-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethyl)pipe...)
Affinity DataIC50: 51nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338437BDBM50338437(methyl 3-(4-((R)-1-amino-2-(2,5-difluorophenyl)eth...)
Affinity DataIC50: 54nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338457BDBM50338457(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 55nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338413BDBM50338413(trans-1-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 57nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338415BDBM50338415(trans-(R)-1-(4-((R)-1-amino-2-(2,5-difluorophenyl)...)
Affinity DataIC50: 70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338429BDBM50338429((R)-2-(2,5-difluorophenyl)-1-(1-(2,6-dimethylpyrid...)
Affinity DataIC50: 71nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338436BDBM50338436((R)-5-(4-(1-amino-2-(2,5-difluorophenyl)ethyl)pipe...)
Affinity DataIC50: 72nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338434BDBM50338434((R)-2-(2,5-difluorophenyl)-1-(1-(pyrimidin-5-yl)pi...)
Affinity DataIC50: 75nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338428BDBM50338428((R)-5-(4-(1-amino-2-(2,5-difluorophenyl)ethyl)pipe...)
Affinity DataIC50: 77nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338435BDBM50338435((R)-2-(2,5-difluorophenyl)-1-(1-(2-methoxypyrimidi...)
Affinity DataIC50: 78nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338431BDBM50338431((R)-ethyl 5-(4-(1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 82nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338448BDBM50338448(trans-4-(N-(4-((R)-1-amino-2-(2,5-difluorophenyl)e...)
Affinity DataIC50: 84nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338443BDBM50338443(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 85nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338451BDBM50338451(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 94nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338447BDBM50338447(trans-3-(N-(4-((R)-1-amino-2-(2,5-difluorophenyl)e...)
Affinity DataIC50: 99nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338455BDBM50338455(trans-N-(5-(N-(4-((R)-1-amino-2-(2,5-difluoropheny...)
Affinity DataIC50: 100nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338405BDBM50338405(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 100nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338430BDBM50338430((R)-2-(2,5-difluorophenyl)-1-(1-(6-fluoropyridin-3...)
Affinity DataIC50: 110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338426BDBM50338426((R)-2-(2,5-difluorophenyl)-1-(1-(pyridin-3-yl)pipe...)
Affinity DataIC50: 110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338467BDBM50338467(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338404BDBM50338404(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338456BDBM50338456(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338473BDBM50338473(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338442BDBM50338442(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338471BDBM50338471(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 120nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338464BDBM50338464(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 120nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338472BDBM50338472(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 120nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338450BDBM50338450(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 130nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338466BDBM50338466(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 130nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338424BDBM50338424((R)-2-(2,5-difluorophenyl)-1-(1-(methylsulfonyl)pi...)
Affinity DataIC50: 130nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338469BDBM50338469(trans-4-((4-((R)-1-amino-2-(2,5-difluorophenyl)eth...)
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338470BDBM50338470(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338445BDBM50338445(trans-4-amino-N-(4-((R)-1-amino-2-(2,5-difluorophe...)
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338441BDBM50338441(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338474BDBM50338474(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338475BDBM50338475(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338449BDBM50338449(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 150nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338454BDBM50338454(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 170nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338440BDBM50338440(trans-N-(4-((S)-1-amino-2-oxo-2-(thiazolidin-3-yl)...)
Affinity DataIC50: 170nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338444BDBM50338444(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 180nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338414BDBM50338414(trans-(S)-1-(4-((R)-1-amino-2-(2,5-difluorophenyl)...)
Affinity DataIC50: 200nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338420BDBM50338420(trans-3-(((4-((R)-1-amino-2-(2,5-difluorophenyl)et...)
Affinity DataIC50: 220nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338476BDBM50338476(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 260nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50338461BDBM50338461(trans-N-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50: 260nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
Displayed 1 to 50 (of 375 total ) | Next | Last >>
Jump to: