Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50033134
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340102(CHEMBL1762820 | N-ethyl-N-(3-fluoropropyl)-8-(6-me...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340103(CHEMBL1762821 | N-(3-fluoropropyl)-8-(6-methoxy-2-...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340101(CHEMBL1762819 | N-(2-fluoroethyl)-8-(6-methoxy-2-m...)
Affinity DataIC50:  5.5nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340100(CHEMBL1762818 | N-ethyl-N-(2-fluoroethyl)-8-(6-met...)
Affinity DataIC50:  5.80nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340104(3-((3-fluoropropyl)(8-(6-methoxy-2-methylpyridin-3...)
Affinity DataIC50:  6.5nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340105(CHEMBL1762823 | N-(3-fluoropropyl)-N-(2-methoxyeth...)
Affinity DataIC50:  35nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340106(CHEMBL1762824 | N-(3-fluoropropyl)-N-(2-methoxyeth...)
Affinity DataIC50:  390nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340107(8-(2,4-dimethoxypyrimidin-5-yl)-N-(3-fluoropropyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed