Compile Data Set for Download or QSAR
Report error Found 100 Enz. Inhib. hit(s) with all data for entry = 50033137
LigandPNGBDBM50340201(N-(3-Chloro-phenyl)-2-[(3R,4S)-1-[2-(1,1-dioxo-hex...)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340188(N-(3-chlorophenyl)-2-((3R,4S)-1-(3,4-dimethoxyphen...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340188(N-(3-chlorophenyl)-2-((3R,4S)-1-(3,4-dimethoxyphen...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340201(N-(3-Chloro-phenyl)-2-[(3R,4S)-1-[2-(1,1-dioxo-hex...)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340204(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340199(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340204(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340197(rac-6-chloro-2-(2-((3R,4S)-1-(3,4-dimethoxypheneth...)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340200(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340200(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340202(N-(3-chlorophenyl)-2-((3R,4S)-1-(2-(4-hydroxytetra...)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340205(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340180(rac-3-chloro-N-(((3S,4S)-1-(4-methoxyphenethyl)-4-...)
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340196(rac-6-chloro-2-(((3R,4S)-1-(3,4-dimethoxyphenethyl...)
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340189(rac-N-(3-chlorophenyl)-2-((3R,4S)-1-(3,4-dimethoxy...)
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340203(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 30nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340176(rac-3-chloro-N-(((3S,4S)-1-(3-(3,4-dimethoxyphenyl...)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340190(rac-N-(3-chlorobenzyl)-2-((3R,4S)-1-(3,4-dimethoxy...)
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340199(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 37nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340188(N-(3-chlorophenyl)-2-((3R,4S)-1-(3,4-dimethoxyphen...)
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340188(N-(3-chlorophenyl)-2-((3R,4S)-1-(3,4-dimethoxyphen...)
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340191(rac-3-chloro-N-(2-((3R,4S)-1-(3,4-dimethoxypheneth...)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340203(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 44nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340198(rac-6-chloro-2-(2-((3R,4S)-1-(3,4-dimethoxypheneth...)
Affinity DataIC50: 45nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340205(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 46nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340179(rac-3-chloro-N-(((3S,4S)-1-(3-methoxyphenethyl)-4-...)
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340191(rac-3-chloro-N-(2-((3R,4S)-1-(3,4-dimethoxypheneth...)
Affinity DataIC50: 56nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340202(N-(3-chlorophenyl)-2-((3R,4S)-1-(2-(4-hydroxytetra...)
Affinity DataIC50: 57nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340188(N-(3-chlorophenyl)-2-((3R,4S)-1-(3,4-dimethoxyphen...)
Affinity DataIC50: 66nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340188(N-(3-chlorophenyl)-2-((3R,4S)-1-(3,4-dimethoxyphen...)
Affinity DataIC50: 66nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340191(rac-3-chloro-N-(2-((3R,4S)-1-(3,4-dimethoxypheneth...)
Affinity DataIC50: 77nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340197(rac-6-chloro-2-(2-((3R,4S)-1-(3,4-dimethoxypheneth...)
Affinity DataIC50: 91nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340153(rac-N-(((3S,4S)-(1-(3,4-dimethoxyphenethyl)-4-(4-m...)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340197(rac-6-chloro-2-(2-((3R,4S)-1-(3,4-dimethoxypheneth...)
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340200(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340145(3-chloro-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl)-4-...)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340145(3-chloro-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl)-4-...)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340163(rac-3-chloro-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl...)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340204(N-(3-chlorophenyl)-2-((3R,4S)-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 140nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340196(rac-6-chloro-2-(((3R,4S)-1-(3,4-dimethoxyphenethyl...)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340145(3-chloro-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl)-4-...)
Affinity DataIC50: 160nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340146(rac-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl)-4-(4-me...)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340145(3-chloro-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl)-4-...)
Affinity DataIC50: 160nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340179(rac-3-chloro-N-(((3S,4S)-1-(3-methoxyphenethyl)-4-...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340164(rac-3-chloro-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340165(rac-3-chloro-N-(((3S,4S)-4-(4-chlorophenyl)-1-(3,4...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340176(rac-3-chloro-N-(((3S,4S)-1-(3-(3,4-dimethoxyphenyl...)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340145(3-chloro-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl)-4-...)
Affinity DataIC50: 250nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340145(3-chloro-N-(((3S,4S)-1-(3,4-dimethoxyphenethyl)-4-...)
Affinity DataIC50: 250nMAssay Description:Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340177(rac-3-chloro-N-(((3S,4S)-1-(4-(3,4-dimethoxyphenyl...)
Affinity DataIC50: 250nMAssay Description:Antagonist activity at MCHR1 by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
Displayed 1 to 50 (of 100 total ) | Next | Last >>
Jump to: