Compile Data Set for Download or QSAR
maximum 50k data
Found 96 Enz. Inhib. hit(s) with all data for entry = 50033157
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340572((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340566(CHEMBL1762535 | N2-(3,5-dimorpholinophenyl)-N4-(5-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340570((2-chloro-5-((2-(3,5-dimorpholinophenylamino)pyrim...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340576(CHEMBL1762525 | N2-(3,5-dimorpholinophenyl)-N4-(3-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340551((3-(isopropyl(2-(3-(methylsulfonyl)-5-morpholinoph...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340555((4-methyl-3-(methyl(2-(3-(methylsulfonyl)-5-morpho...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340571((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340562((4-methyl-3-(methyl(2-(3-(4-methylpiperazin-1-yl)-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340554((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340556((3-((2-(3-methoxy-5-morpholinophenylamino)pyrimidi...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340553((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340560((4-methyl-3-(methyl(2-(3-morpholino-5-(morpholinom...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340567(CHEMBL1762534 | N2-(3,5-dimorpholinophenyl)-N4-(6-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340577(CHEMBL1762524 | N4-(3-chlorophenyl)-N2-(3,5-dimorp...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340572((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340561(4-(3-(4-((5-(hydroxymethyl)-2-methylphenyl)(methyl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340551((3-(isopropyl(2-(3-(methylsulfonyl)-5-morpholinoph...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340550((3-((2-(2,6-dimorpholinopyridin-4-ylamino)pyrimidi...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340557((3-((2-(3-(2-methoxyethoxy)-5-morpholinophenylamin...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340558((4-methyl-3-(methyl(2-(3-morpholino-5-(tetrahydro-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340578(CHEMBL1762523 | N2-(3,5-dimorpholinophenyl)-N4-met...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340563((4-methyl-3-(methyl(2-(3-morpholino-5-(1,4-oxazepa...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340573((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340576(CHEMBL1762525 | N2-(3,5-dimorpholinophenyl)-N4-(3-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340564((4-methyl-3-(methyl(2-(3-morpholino-5-(piperidin-1...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340574(CHEMBL1762527 | N2-(3,5-dimorpholinophenyl)-N4-(5-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340579(CHEMBL1762522 | N2-(3,5-dimorpholinophenyl)-N4-met...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340564((4-methyl-3-(methyl(2-(3-morpholino-5-(piperidin-1...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340555((4-methyl-3-(methyl(2-(3-(methylsulfonyl)-5-morpho...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340577(CHEMBL1762524 | N4-(3-chlorophenyl)-N2-(3,5-dimorp...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340571((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340552((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340552((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340553((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340568(CHEMBL1762533 | N2-(3,5-dimorpholinophenyl)-N4-(4-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340570((2-chloro-5-((2-(3,5-dimorpholinophenylamino)pyrim...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340550((3-((2-(2,6-dimorpholinopyridin-4-ylamino)pyrimidi...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340554((3-((2-(3,5-dimorpholinophenylamino)pyrimidin-4-yl...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340549((3-((2-(2,6-dimorpholinopyrimidin-4-ylamino)pyrimi...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340565((4-methyl-3-(methyl(2-(3-morpholino-5-(pyrrolidin-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340580(CHEMBL1762521 | N2-(3,5-dimorpholinophenyl)-N4-met...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340559((3-(4-((5-(hydroxymethyl)-2-methylphenyl)(methyl)a...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340575(CHEMBL1762526 | N4-(2,5-dimethylphenyl)-N2-(3,5-di...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340574(CHEMBL1762527 | N2-(3,5-dimorpholinophenyl)-N4-(5-...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340570((2-chloro-5-((2-(3,5-dimorpholinophenylamino)pyrim...)
Affinity DataIC50:  22nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340558((4-methyl-3-(methyl(2-(3-morpholino-5-(tetrahydro-...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340560((4-methyl-3-(methyl(2-(3-morpholino-5-(morpholinom...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340565((4-methyl-3-(methyl(2-(3-morpholino-5-(pyrrolidin-...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340577(CHEMBL1762524 | N4-(3-chlorophenyl)-N2-(3,5-dimorp...)
Affinity DataIC50:  27nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340578(CHEMBL1762523 | N2-(3,5-dimorpholinophenyl)-N4-met...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human EphB4 autophosphorylation expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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