Compile Data Set for Download or QSAR
Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 50033386
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344294BDBM50344294((R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-3-ylmeth...)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344287BDBM50344287((R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-phenylprop...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344292BDBM50344292((R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-2-ylmeth...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344270BDBM50344270((R)-quinuclidin-3-yl phenyl(thiophen-2-ylmethyl)ca...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344271BDBM50344271((R)-quinuclidin-3-yl phenyl(thiophen-3-ylmethyl)ca...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344292BDBM50344292((R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-2-ylmeth...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344303BDBM50344303((R)-quinuclidin-3-yl benzyl(phenyl)carbamate | CHE...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344294BDBM50344294((R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-3-ylmeth...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344291BDBM50344291((R)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-...)
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344301BDBM50344301((R)-3-((3-fluorophenyl)(3,4,5-trifluorobenzyl)carb...)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344297BDBM50344297((R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-(thiophen-2...)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344293BDBM50344293((R)-3-(phenyl(thiophen-3-ylmethyl)carbamoyloxy)-1-...)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344288BDBM50344288((R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-(thiophen-...)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344270BDBM50344270((R)-quinuclidin-3-yl phenyl(thiophen-2-ylmethyl)ca...)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344296BDBM50344296((R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-phenylpropy...)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344298BDBM50344298((R)-3-(butyl(phenyl)carbamoyloxy)-1-(2-phenoxyethy...)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344278BDBM50344278((R)-quinuclidin-3-yl butyl(thiophen-2-ylmethyl)car...)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344274BDBM50344274((R)-quinuclidin-3-yl pentyl(phenyl)carbamate | CHE...)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344283BDBM50344283((R)-quinuclidin-3-yl 3-fluorophenyl(3,4,5-trifluor...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344299BDBM50344299((R)-1-(3-phenylpropyl)-3-(m-tolyl(2,4,5-trifluorob...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344269BDBM50344269((R)-quinuclidin-3-yl phenethyl(phenyl)carbamate | ...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344282BDBM50344282((R)-quinuclidin-3-yl m-tolyl(2,4,5-trifluorobenzyl...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344289BDBM50344289((R)-3-(benzyl(phenyl)carbamoyloxy)-1-(2-phenoxyeth...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344271BDBM50344271((R)-quinuclidin-3-yl phenyl(thiophen-3-ylmethyl)ca...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344301BDBM50344301((R)-3-((3-fluorophenyl)(3,4,5-trifluorobenzyl)carb...)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344292BDBM50344292((R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-2-ylmeth...)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344273BDBM50344273((R)-quinuclidin-3-yl butyl(phenyl)carbamate | CHEM...)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344300BDBM50344300((R)-1-(2-phenoxyethyl)-3-(m-tolyl(2,4,5-trifluorob...)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344303BDBM50344303((R)-quinuclidin-3-yl benzyl(phenyl)carbamate | CHE...)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344282BDBM50344282((R)-quinuclidin-3-yl m-tolyl(2,4,5-trifluorobenzyl...)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344298BDBM50344298((R)-3-(butyl(phenyl)carbamoyloxy)-1-(2-phenoxyethy...)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344288BDBM50344288((R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-(thiophen-...)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344283BDBM50344283((R)-quinuclidin-3-yl 3-fluorophenyl(3,4,5-trifluor...)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344287BDBM50344287((R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-phenylprop...)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344281BDBM50344281((R)-quinuclidin-3-yl 3-fluorobenzyl(3-fluorophenyl...)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344294BDBM50344294((R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-3-ylmeth...)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344291BDBM50344291((R)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-...)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344274BDBM50344274((R)-quinuclidin-3-yl pentyl(phenyl)carbamate | CHE...)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344289BDBM50344289((R)-3-(benzyl(phenyl)carbamoyloxy)-1-(2-phenoxyeth...)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344270BDBM50344270((R)-quinuclidin-3-yl phenyl(thiophen-2-ylmethyl)ca...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344297BDBM50344297((R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-(thiophen-2...)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344293BDBM50344293((R)-3-(phenyl(thiophen-3-ylmethyl)carbamoyloxy)-1-...)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344300BDBM50344300((R)-1-(2-phenoxyethyl)-3-(m-tolyl(2,4,5-trifluorob...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344281BDBM50344281((R)-quinuclidin-3-yl 3-fluorobenzyl(3-fluorophenyl...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344277BDBM50344277((R)-quinuclidin-3-yl bis(thiophen-2-ylmethyl)carba...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344296BDBM50344296((R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-phenylpropy...)
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344285BDBM50344285(quinuclidin-4-yl biphenyl-2-ylcarbamate hydrochlor...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344299BDBM50344299((R)-1-(3-phenylpropyl)-3-(m-tolyl(2,4,5-trifluorob...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344291BDBM50344291((R)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-...)
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344269BDBM50344269((R)-quinuclidin-3-yl phenethyl(phenyl)carbamate | ...)
Affinity DataIC50: 3.60nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
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